SCHEMBL5205062

SCHEMBL5205062

Cc1ccc(F)c(C(=O)N2CCC(c3cn(Cc4ccc(C#N)cc4)c4ccccc34)C2)c1Cl

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMO Q99835 1/20 0.46
CNR2 P34972 1/20 0.44
LMNA P02545 2/20 0.43
HTT P42858 2/20 0.43
SLC2A1 P11166 1/20 0.42
KDM1A O60341 3/20 0.42
POLB P06746 1/20 0.41
NPSR1 Q6W5P4 2/20 0.40
MAPT P10636 2/20 0.40
HDAC3 O15379 1/20 0.40
HDAC1 Q13547 1/20 0.40
HDAC2 Q92769 1/20 0.40
HDAC10 Q969S8 1/20 0.40
HDAC8 Q9BY41 1/20 0.40
HDAC6 Q9UBN7 1/20 0.40
NCOR2 Q9Y618 1/20 0.40
HRH2 P25021 1/20 0.39
PTGS2 P35354 1/20 0.39
CCR3 P51677 1/20 0.39
SLC5A1 P13866 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4859112 0.81 RORC (0.47) LMNAPOLBNPSR1MAPTALDH1A1
SCHEMBL5203814 0.79 SMO (0.51) SMOCNR2LMNAHTTSLC2A1
SCHEMBL5487349 0.78 ADAM17 (0.36) SMOLMNAHTTPOLBALDH1A1
SCHEMBL5202142 0.78 LMNA (0.50) SMOCNR2LMNAHTTSLC2A1
SCHEMBL3598410 0.78 SMO (0.54) SMOCNR2LMNAHTTSLC2A1
SCHEMBL5204299 0.77 SLC5A1 (0.47) LMNAHTTSLC2A1NPSR1HDAC3
SCHEMBL5204484 0.77 SLC2A1 (0.47) LMNAHTTSLC2A1NPSR1MAPT
SCHEMBL5206978 0.75 SLC5A1 (0.49) LMNAHTTSLC2A1NPSR1HDAC3
SCHEMBL5206068 0.75 LMNA (0.49) SMOCNR2LMNAHTTSLC2A1
SCHEMBL5201634 0.75 SLC2A1 (0.47) SMOCNR2LMNAHTTSLC2A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1654253-B1 SUBSTITUTED 3-PYRROLIDIN-INDOLE DERIVATIVES GRUENENTHAL GMBH (DE) 2007-01-03 EP claimed
EP-1654253-B1 SUBSTITUTED 3-PYRROLIDIN-INDOLE DERIVATIVES GRUENENTHAL GMBH (DE) 2007-01-03 EP disclosed