SCHEMBL5203814

SCHEMBL5203814

COCC(=O)N1CCC(c2cn(Cc3ccc(C#N)cc3)c3ccccc23)C1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMO Q99835 1/20 0.51
CNR2 P34972 2/20 0.49
LMNA P02545 3/20 0.48
HTT P42858 3/20 0.48
CYP3A4 P08684 1/20 0.48
POLB P06746 1/20 0.45
NPSR1 Q6W5P4 2/20 0.44
HRH2 P25021 1/20 0.44
MAPT P10636 1/20 0.44
HDAC3 O15379 1/20 0.44
HDAC1 Q13547 1/20 0.44
HDAC2 Q92769 1/20 0.44
HDAC10 Q969S8 1/20 0.44
HDAC8 Q9BY41 1/20 0.44
HDAC6 Q9UBN7 1/20 0.44
NCOR2 Q9Y618 1/20 0.44
KDM1A O60341 2/20 0.42
HTR2A P28223 2/20 0.42
HTR2C P28335 2/20 0.42
HTR2B P41595 2/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5202142 0.83 LMNA (0.50) SMOCNR2LMNAHTTPOLB
SCHEMBL4852934 0.82 HRH2 (0.50) LMNAHTTPOLBNPSR1HRH2
SCHEMBL5206068 0.82 LMNA (0.49) SMOCNR2LMNAHTTCYP3A4
SCHEMBL5205062 0.79 SMO (0.46) SMOCNR2LMNAHTTPOLB
SCHEMBL4859500 0.78 KMT2A (0.52) SMOLMNAHTTCYP3A4POLB
SCHEMBL3598410 0.78 SMO (0.54) SMOCNR2LMNAHTTCYP3A4
SCHEMBL5203146 0.77 SMO (0.47) SMOCNR2LMNAHTTPOLB
SCHEMBL5203143 0.74 CNR2 (0.43) SMOCNR2LMNAHTTPOLB
SCHEMBL5204486 0.74 MAPT (0.54) LMNAHTTNPSR1HRH2MAPT
SCHEMBL13445248 0.73 SMO (0.57) SMOCNR2CYP3A4NPSR1HRH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1654253-B1 SUBSTITUTED 3-PYRROLIDIN-INDOLE DERIVATIVES GRUENENTHAL GMBH (DE) 2007-01-03 EP claimed
EP-1654253-B1 SUBSTITUTED 3-PYRROLIDIN-INDOLE DERIVATIVES GRUENENTHAL GMBH (DE) 2007-01-03 EP disclosed