SCHEMBL5204889

SCHEMBL5204889

CC(C)(C)OC(=O)NCc1ccc(Oc2ccccc2N(Cc2ccc(-c3ccccc3)cc2)C(=O)CCC(=O)O)cc1

nearest known ligand 0.47

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 2/20 0.47
SDCBP O00560 1/20 0.41
SDC2 P34741 1/20 0.41
LTB4R2 Q9NPC1 1/20 0.39
TSPO P30536 3/20 0.38
ALDH1A1 P00352 1/20 0.38
NPC1 O15118 1/20 0.38
RAB9A P51151 1/20 0.38
NAMPT P43490 1/20 0.38
CTSS P25774 1/20 0.38
CTSK P43235 1/20 0.38
AKT1 P31749 2/20 0.37
KMT2A Q03164 2/20 0.36
LTA4H P09960 1/20 0.36
MEN1 O00255 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5208000 0.91 HDAC1 (0.44) HDAC1SDCBPSDC2TSPOAKT1
SCHEMBL5206192 0.88 HDAC1 (0.40) HDAC1SDCBPSDC2TSPOALDH1A1
SCHEMBL5202825 0.83 HDAC1 (0.44) HDAC1SDCBPSDC2LTB4R2CTSS
SCHEMBL5205381 0.83 HDAC1 (0.41) HDAC1SDCBPSDC2TSPO
SCHEMBL5204311 0.80 ALDH1A1 (0.42) HDAC1SDCBPSDC2TSPOALDH1A1
SCHEMBL5204997 0.78 ALDH1A1 (0.43) HDAC1TSPOALDH1A1RAB9ACTSS
SCHEMBL5202464 0.78 ALDH1A1 (0.41) HDAC1TSPOALDH1A1
SCHEMBL5208677 0.77 NR3C1 (0.41) HDAC1TSPOALDH1A1KMT2A
SCHEMBL7242557 0.76 HDAC1 (0.50) HDAC1SDCBPSDC2NAMPTCTSS
SCHEMBL1691047 0.76 HDAC1 (0.67) HDAC1SDCBPSDC2ALDH1A1NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7160887-B1 Aromatic amine derivatives, their production and use TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2007-01-09 US disclosed