SCHEMBL5212799

SCHEMBL5212799

CN1CCC(C(=O)c2cccc(NS(C)(=O)=O)c2)CC1

nearest known ligand 0.61

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
HTR1F P30939 4/20 0.61
ALDH1A1 P00352 1/20 0.56
SMN1; SMN2 Q16637 1/20 0.56
POLB P06746 2/20 0.53
NPSR1 Q6W5P4 1/20 0.52
KCNH2 Q12809 2/20 0.50
CYP3A4 P08684 2/20 0.50
CYP2C19 P33261 2/20 0.50
CYP2D6 P10635 1/20 0.50
KDM4E B2RXH2 2/20 0.49
DHX9 Q08211 1/20 0.46
MEN1 O00255 3/20 0.46
KMT2A Q03164 3/20 0.46
HPGD P15428 1/20 0.45
CYP1A2 P05177 1/20 0.45
PRMT5 O14744 2/20 0.44
FKBP1A P62942 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5213124 0.85 HTR1F (0.56) HTR1FALDH1A1POLBMEN1KMT2A
SCHEMBL5210617 0.84 HTR1F (0.66) HTR1FNPSR1CYP2C19MEN1KMT2A
SCHEMBL5210461 0.83 HTR1F (0.60) HTR1FPOLBNPSR1CYP2C19MEN1
SCHEMBL5212363 0.83 TCF4 (0.59) HTR1FALDH1A1SMN1; SMN2POLBNPSR1
Hydrochloric Acid SCHEMBL9444478 0.83 KCNH2 (0.60) HTR1FALDH1A1POLBKCNH2CYP3A4
SCHEMBL5213302 0.83 HTR1F (0.65) HTR1FNPSR1CYP2C19MEN1KMT2A
Hydrochloric Acid SCHEMBL9444456 0.83 KCNH2 (0.60) HTR1FALDH1A1POLBKCNH2CYP3A4
SCHEMBL5210686 0.83 HTR1F (0.53) HTR1FALDH1A1SMN1; SMN2NPSR1MEN1
SCHEMBL5208596 0.83 HTR1F (0.53) HTR1FALDH1A1SMN1; SMN2POLBNPSR1
SCHEMBL5210843 0.83 ITGA1 (0.58) HTR1FALDH1A1SMN1; SMN2POLBKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1153013-B1 5-HT1F AGONISTS LILLY CO ELI (US) 2007-10-31 EP disclosed
EP-1153013-B1 5-HT1F AGONISTS LILLY CO ELI (US) 2007-10-31 EP disclosed
US-6777428-B1 INHIBIT PEPTIDE EXTRAVASATION DUE TO STIMULATION OF THE TRIGEMINAL GANGLIA, AND ARE THEREFORE USEFUL FOR THE TREATMENT OF MIGRAINE AND ASSOCIATED DISORDERS ELI LILLY AND COMPANY 2004-08-17 US disclosed
CN-1149195-C 5-HTIF agonists 2004-05-12 CN disclosed
EP-1153013-A2 5-HT1F AGONISTS ELI LILLY AND COMPANY (US) 2001-11-14 EP disclosed
WO-2000047559-A2 5-HT1F AGONISTS ELI LILLY AND COMPANY (US) 2000-08-17 WO disclosed