SCHEMBL5212995

SCHEMBL5212995

CCCN1CCN(S(=O)(=O)CCCN2CCC(C)CC2)CC1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR4 Q13639 3/20 0.45
KDM4E B2RXH2 4/20 0.45
ALDH1A1 P00352 3/20 0.45
NPC1 O15118 1/20 0.40
RAB9A P51151 1/20 0.40
ALOX15 P16050 2/20 0.39
POLB P06746 1/20 0.39
SIGMAR1 Q99720 3/20 0.38
CARM1 Q86X55 1/20 0.38
PRMT6 Q96LA8 1/20 0.38
PRMT1 Q99873 1/20 0.38
PRMT8 Q9NR22 1/20 0.38
DRD2 P14416 1/20 0.37
GNAI3 P08754 1/20 0.37
GNAO1 P09471 1/20 0.37
GNAI1 P63096 1/20 0.37
HTR7 P34969 1/20 0.37
CYP1A2 P05177 1/20 0.37
CYP2D6 P10635 1/20 0.37
CYP2C19 P33261 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5212984 0.87 HTR4 (0.45) HTR4KDM4EALDH1A1ALOX15SIGMAR1
SCHEMBL5216687 0.84 HTR4 (0.48) HTR4KDM4EALOX15SIGMAR1DRD2
SCHEMBL5215065 0.84 HTR4 (0.49) HTR4KDM4EALDH1A1NPC1RAB9A
SCHEMBL5213629 0.82 HTR4 (0.47) HTR4KDM4EALDH1A1ALOX15POLB
SCHEMBL5216679 0.82 SMN1; SMN2 (0.49) HTR4KDM4EALDH1A1NPC1RAB9A
SCHEMBL14375265 0.82 HTR4 (0.45) HTR4ALDH1A1RAB9ACARM1PRMT6
SCHEMBL13411085 0.79 ALDH1A1 (0.50) KDM4EALDH1A1NPC1RAB9AALOX15
SCHEMBL5219353 0.78 HTR4 (0.46) HTR4KDM4EALDH1A1RAB9AALOX15
SCHEMBL5215771 0.77 HTR4 (0.47) HTR4KDM4EALDH1A1ALOX15CYP1A2
SCHEMBL10263618 0.76 MEN1 (0.47) KDM4EPOLBSIGMAR1DRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1112270-B1 DIHYDROBENZODIOXINE CARBOXAMIDE AND KETONE DERIVATIVES AS 5-HT4 RECEPTOR ANTAGONISTS HOFFMANN LA ROCHE (CH) 2007-03-21 EP claimed