SCHEMBL5216679

SCHEMBL5216679

CCCN1CCN(S(=O)(=O)CCCN2CCC(C(N)=O)CC2)CC1

nearest known ligand 0.49

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 3/20 0.49
HTR4 Q13639 3/20 0.46
ALDH1A1 P00352 4/20 0.46
GAA P10253 1/20 0.46
ALOX15 P16050 1/20 0.45
BCHE P06276 1/20 0.42
NPC1 O15118 2/20 0.41
LMNA P02545 3/20 0.40
DRD2 P14416 1/20 0.40
HRH1 P35367 1/20 0.40
DRD3 P35462 1/20 0.40
KDM4E B2RXH2 2/20 0.39
HTT P42858 1/20 0.39
CYP1A2 P05177 2/20 0.39
CYP2C9 P11712 1/20 0.39
RAB9A P51151 1/20 0.39
CYP2D6 P10635 1/20 0.39
CYP2C19 P33261 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5215761 0.93 ALOX15 (0.52) SMN1; SMN2HTR4ALDH1A1GAAALOX15
SCHEMBL5215957 0.92 SMN1; SMN2 (0.60) SMN1; SMN2HTR4ALDH1A1GAAALOX15
SCHEMBL5212302 0.89 SMN1; SMN2 (0.50) SMN1; SMN2HTR4ALDH1A1GAAALOX15
SCHEMBL5216773 0.86 SMN1; SMN2 (0.42) SMN1; SMN2HTR4ALDH1A1GAAALOX15
SCHEMBL5219357 0.86 HTR4 (0.50) SMN1; SMN2HTR4ALDH1A1GAAALOX15
SCHEMBL5217099 0.85 HTR4 (0.48) SMN1; SMN2HTR4ALDH1A1GAAALOX15
SCHEMBL5214681 0.84 HTR4 (0.46) SMN1; SMN2HTR4ALDH1A1GAAALOX15
SCHEMBL5306262 0.83 HTR4 (0.46) SMN1; SMN2HTR4ALDH1A1GAAALOX15
SCHEMBL5212995 0.82 HTR4 (0.45) SMN1; SMN2HTR4ALDH1A1ALOX15NPC1
SCHEMBL5216687 0.81 HTR4 (0.48) HTR4ALOX15DRD2KDM4ECYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1112270-B1 DIHYDROBENZODIOXINE CARBOXAMIDE AND KETONE DERIVATIVES AS 5-HT4 RECEPTOR ANTAGONISTS HOFFMANN LA ROCHE (CH) 2007-03-21 EP claimed