SCHEMBL5213274

SCHEMBL5213274

NS(=O)(=O)Cc1ccc2ncccc2c1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.50
MAPT P10636 2/20 0.50
KDM4E B2RXH2 1/20 0.50
TP53 P04637 1/20 0.50
HSP90AA1 P07900 1/20 0.50
HSP90AB1 P08238 1/20 0.50
TSHR P16473 1/20 0.50
CASP1 P29466 1/20 0.50
HTT P42858 1/20 0.50
ATM Q13315 1/20 0.50
SMN1; SMN2 Q16637 1/20 0.50
HSD17B10 Q99714 1/20 0.50
NPC1 O15118 3/20 0.49
POLB P06746 2/20 0.49
RAB9A P51151 1/20 0.49
HDAC3 O15379 2/20 0.48
DAO P14920 1/20 0.47
DYRK1A Q13627 1/20 0.44
MET P08581 4/20 0.44
CHKA P35790 2/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL27681462 0.98 ALDH1A1 (0.49) ALDH1A1MAPTKDM4ETP53HSP90AA1
SCHEMBL29673226 0.78 ALDH1A1 (0.58) ALDH1A1MAPTKDM4ETP53HSP90AA1
SCHEMBL507149 0.78 ALDH1A1 (0.58) ALDH1A1MAPTKDM4ETP53HSP90AA1
SCHEMBL2107923 0.78 NPC1 (0.57) ALDH1A1MAPTKDM4ETP53HSP90AA1
SCHEMBL30586439 0.78 ALDH1A1 (0.58) ALDH1A1MAPTKDM4ETP53HSP90AA1
Iodide SCHEMBL20524052 0.76 ALDH1A1 (0.56) ALDH1A1MAPTKDM4ETP53HSP90AA1
SCHEMBL1764709 0.75 CA1 (0.57) CA1CA2CA5ACA9
SCHEMBL6383861 0.75 CA2 (0.37) METCA1CA2CA5ACA9
SCHEMBL6961498 0.75 DAO (0.57) ALDH1A1MAPTKDM4ETP53HSP90AA1
SCHEMBL2597877 0.75 ALDH1A1 (0.59) ALDH1A1MAPTKDM4ETP53HSP90AA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101039931-A Novel product, method and intermediates for the preparation of azetidine derivatives AVENTIS PHARMA SA (FR) 2007-09-19 CN disclosed
EP-1805167-A2 NOVEL PRODUCT, METHOD AND INTERMEDIATES FOR THE PREPARATION OF AZETIDINE DERIVATIVES Aventis Pharma S.A. (FR) 2007-07-11 EP disclosed
WO-2006040465-A2 NOVEL PRODUCT, METHOD AND INTERMEDIATES FOR THE PREPARATION OF AZETIDINE DERIVATIVES AVENTIS PHARMA S.A. (FR) 2006-04-20 WO disclosed