SCHEMBL1764709

SCHEMBL1764709

NS(=O)(=O)Cc1ccc2ccccc2c1

nearest known ligand 0.57

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CA1 P00915 8/20 0.57
CA2 P00918 8/20 0.57
CA9 Q16790 6/20 0.57
CA5A P35218 1/20 0.57
LMNA P02545 1/20 0.52
CYP1A2 P05177 2/20 0.50
CYP2A6 P11509 1/20 0.50
CA12 O43570 2/20 0.49
CA4 P22748 2/20 0.49
CA7 P43166 2/20 0.49
HTR2A P28223 1/20 0.47
HTR2C P28335 1/20 0.47
HTR2B P41595 1/20 0.47
PTGES2 Q9H7Z7 1/20 0.47
MC4R P32245 1/20 0.44
MC5R P33032 1/20 0.44
TEAD4 Q15561 1/20 0.43
MLNR O43193 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27450675 0.83 CYP1A2 (0.54) CA1CA2CA9LMNACYP1A2
SCHEMBL9464709 0.82 CA2 (0.45) CA1CA2CA9CA5ACA12
SCHEMBL294031 0.82 CYP1A2 (0.52) CA1CA2CA9LMNACYP1A2
SCHEMBL23722235 0.81 PTGES2 (0.58) CA1CA2CA9LMNACYP1A2
SCHEMBL30647960 0.81 PTGES2 (0.58) CA1CA2CA9LMNACYP1A2
SCHEMBL11692490 0.81 CA2 (0.44) CA1CA2CA9CA5ACA12
SCHEMBL17374931 0.81 CA2 (0.48) CA1CA2CA9CA5ACYP2A6
SCHEMBL12230567 0.80 CYP1A2 (0.50) CA1CA2CA9LMNACYP1A2
SCHEMBL171848 0.80 CYP1A2 (0.55) LMNACYP1A2CYP2A6HTR2AHTR2C
SCHEMBL2374771 0.80 CYP1A2 (0.50) CA1CA2CA9LMNACYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021114313-A1 ION CHANNEL ANTAGONISTS/BLOCKERS AND USES THEREOF SHANGHAI EAST HOSPITAL (CN) 2021-06-17 WO disclosed
EP-2513092-A1 HETEROCYCLIC ANTIVIRAL COMPOUNDS F. Hoffmann-La Roche AG (CH) 2012-10-24 EP disclosed
WO-2011073114-A1 HETEROCYCLIC ANTIVIRAL COMPOUNDS F. HOFFMANN-LA ROCHE AG (CH) 2011-06-23 WO disclosed
US-20110123490-A1 HETEROCYCLIC ANTIVIRAL COMPOUNDS ROCHE PALO ALTO LLC (US) 2011-05-26 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110123490-A1 HETEROCYCLIC ANTIVIRAL COMPOUNDS RRM2B, POLR2A, RRM2 CA1 4778/4885CA2 4785/4885CA9 3584/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.