SCHEMBL5214760

SCHEMBL5214760

OCCOc1cccc(Cl)n1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDK9 P50750 1/20 0.41
DYRK1A Q13627 1/20 0.41
DYRK2 Q92630 1/20 0.41
ALDH1A1 P00352 2/20 0.41
RECQL P46063 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.38
HTR7 P34969 2/20 0.38
THRB P10828 1/20 0.37
KMT2A Q03164 1/20 0.37
DRD4 P21917 1/20 0.36
HTR1A P08908 1/20 0.36
ADRA1A P35348 1/20 0.36
CYP3A4 P08684 1/20 0.35
TSHR P16473 1/20 0.35
GPR52 Q9Y2T5 1/20 0.35
HDAC1 Q13547 1/20 0.34
HDAC6 Q9UBN7 1/20 0.34
HDAC5 Q9UQL6 1/20 0.34
F2 P00734 1/20 0.34
CYP11B1 P15538 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15532864 0.89 CDK9 (0.37) CDK9DYRK1ADYRK2L3MBTL1HTR7
SCHEMBL9253185 0.87 CNR2 (0.37) CDK9DYRK1ADYRK2ALDH1A1L3MBTL1
SCHEMBL24343308 0.86 ALDH1A1 (0.54) ALDH1A1RECQLHTR7THRBKMT2A
SCHEMBL13822632 0.81 HTR1B (0.42) CDK9DYRK1ADYRK2L3MBTL1HTR7
SCHEMBL10910803 0.81 MCHR1 (0.42) CDK9DYRK1ADYRK2ALDH1A1L3MBTL1
SCHEMBL5214757 0.81 CYP3A4 (0.39) CDK9DYRK1ADYRK2ALDH1A1L3MBTL1
SCHEMBL10911295 0.79 MCHR1 (0.44) CDK9DYRK1ADYRK2ALDH1A1L3MBTL1
SCHEMBL30328346 0.79 TSHR (0.41) CDK9DYRK1ADYRK2ALDH1A1L3MBTL1
SCHEMBL17980783 0.79 TSHR (0.41) CDK9DYRK1ADYRK2ALDH1A1L3MBTL1
Ammonia Solution, Strong SCHEMBL2186005 0.79 MCHR1 (0.41) CDK9DYRK1ADYRK2ALDH1A1L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2025137541-A1 KINASE MODULATORS AND METHODS OF USE THEREOF NEURON23, INC. (US) 2025-06-26 WO disclosed
EP-1453492-B1 USE OF QUINAZOLINES TO TREAT T-CELL MEDIATED DISEASES ASTRAZENECA AB (SE) 2007-01-24 EP disclosed
US-7157467-B2 Administering compound such as 6-methoxy-4-(2,3-methylenedioxyanilino)-7-(3-morpholinopropoxy)quinazoline for therapy of an autoimmune disease or medical condition selected from transplant rejection and rheumatoid arthritis ASTRAZENECA AB (SE) 2007-01-02 US disclosed
US-7115615-B2 Quinazoline derivatives ASTRAZENECA (SE) 2006-10-03 US disclosed
US-20050014773-A1 Therapeutic use ASTRAZENACA AB (SE) 2005-01-20 US disclosed
EP-1453492-A2 USE OF QUINAZOLINES TO TREAT T-CELL MEDIATED DISEASES Astrazeneca AB (SE) 2004-09-08 EP disclosed
WO-2003045364-A2 USE OF QUINAZOLINES TO TREAT T-CELL MEDIATED DISEASES ASTRAZENECA AB (SE) 2003-06-05 WO disclosed
EP-1313727-A1 QUINAZOLINE DERIVATIVES AstraZeneca AB (SE) 2003-05-28 EP disclosed
WO-2002016352-A1 QUINAZOLINE DERIVATIVES ASTRAZENECA AB (SE) 2002-02-28 WO disclosed
US-4588816-A Preparation of (2-(6-substituted)-pyridinyloxy)alkanols from 2-(6-substituted)pyridinols and organic carbonates THE DOW CHEMICAL COMPANY (US) 1986-05-13 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050014773-A1 Therapeutic use CD4, HLA-DRB1, CD74 CDK9 2999/4885DYRK1A 2843/4885DYRK2 2541/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.