SCHEMBL5215111

SCHEMBL5215111

CN1CCN(S(=O)(=O)CCCN2CCC(CCC(N)=O)CC2)CC1

nearest known ligand 0.46

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
HTR4 Q13639 16/20 0.46
ALDH1A1 P00352 1/20 0.36
ATM Q13315 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5215119 0.83 HTR4 (0.44) HTR4ALDH1A1
SCHEMBL5212302 0.82 SMN1; SMN2 (0.50) HTR4ALDH1A1
SCHEMBL5212310 0.81 NCF1 (0.49) HTR4
SCHEMBL5219357 0.77 HTR4 (0.50) HTR4ALDH1A1
SCHEMBL6855190 0.76 NCF1 (0.48) HTR4ALDH1A1ATM
Bromide SCHEMBL5227189 0.76 HTR4 (0.51) HTR4ALDH1A1
Hydrochloric Acid SCHEMBL30412623 0.74 GNAI3 (0.50) HTR4ALDH1A1ATM
SCHEMBL5219363 0.73 HTR4 (0.48) HTR4ALDH1A1
SCHEMBL5215761 0.73 ALOX15 (0.52) HTR4ALDH1A1
SCHEMBL2429930 0.73 GNAI3 (0.42) HTR4ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1112270-B1 DIHYDROBENZODIOXINE CARBOXAMIDE AND KETONE DERIVATIVES AS 5-HT4 RECEPTOR ANTAGONISTS HOFFMANN LA ROCHE (CH) 2007-03-21 EP disclosed