SCHEMBL5217026

SCHEMBL5217026

COc1cc(CCOc2cccc(F)c2C#N)cc(OC)c1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAOB P27338 1/20 0.42
NPC1 O15118 1/20 0.40
RAB9A P51151 1/20 0.40
ABCB1 P08183 3/20 0.39
FGFR2 P21802 1/20 0.39
FGFR3 P22607 1/20 0.39
LMNA P02545 1/20 0.39
MAPT P10636 1/20 0.39
TSHR P16473 1/20 0.39
HTT P42858 1/20 0.39
TDP1 Q9NUW8 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
SQOR Q9Y6N5 1/20 0.38
PRKACA P17612 1/20 0.38
PRKACG P22612 1/20 0.38
PRKACB P22694 1/20 0.38
CYP1A2 P05177 2/20 0.38
CYP3A4 P08684 2/20 0.38
KDM4E B2RXH2 1/20 0.38
MEN1 O00255 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5219798 0.91 TAAR1 (0.48) MAOBABCB1TDP1SQORKDM4E
SCHEMBL5222695 0.84 MAPK14 (0.40) NPC1RAB9ALMNAMAPTTSHR
SCHEMBL5217387 0.82 CASR (0.41) MAOBNPC1RAB9ALMNAMAPT
SCHEMBL1154474 0.81 CYP11B1 (0.43) NPC1RAB9ALMNAMAPTTSHR
SCHEMBL5224566 0.80 MAPK14 (0.47) MAOBNPC1LMNAMAPTTSHR
SCHEMBL1154302 0.80 LMNA (0.43) MAOBNPC1RAB9ALMNAMAPT
SCHEMBL5225071 0.80 CASR (0.51) LMNAMAPTTSHRHTTCYP2D6
SCHEMBL5220371 0.78 HTR2C (0.44) MAOBNPC1RAB9ACYP1A2CYP3A4
SCHEMBL1154627 0.78 SQOR (0.45) NPC1RAB9ALMNAMAPTTSHR
SCHEMBL5216704 0.78 MAPT (0.42) NPC1RAB9ALMNAMAPTTSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1765810-A1 2,4-DIAMINOQUINAZOLINES FOR SPINAL MUSCULAR ATROPHY Decode Chemistry, Inc. (US) 2007-03-28 EP disclosed
WO-2005123724-A1 2,4-DIAMINOQUINAZOLINES FOR SPINAL MUSCULAR ATROPHY DECODE CHEMISTRY, INC. (US) 2005-12-29 WO disclosed