SCHEMBL5219798

SCHEMBL5219798

COc1cccc(CCOc2cccc(F)c2C#N)c1

nearest known ligand 0.48

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
TAAR1 Q96RJ0 1/20 0.48
ABCB1 P08183 11/20 0.45
HTR1A P08908 2/20 0.45
DRD2 P14416 2/20 0.45
MAOB P27338 1/20 0.44
HTR2C P28335 1/20 0.43
SLC6A4 P31645 1/20 0.43
HTR2B P41595 1/20 0.43
CHRM2 P08172 1/20 0.43
CHRM1 P11229 1/20 0.43
CHRM3 P20309 1/20 0.43
KDM4E B2RXH2 1/20 0.42
MEN1 O00255 1/20 0.42
ALDH1A1 P00352 1/20 0.42
KMT2A Q03164 1/20 0.42
TDP1 Q9NUW8 1/20 0.42
SQOR Q9Y6N5 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5217026 0.91 MAOB (0.42) ABCB1MAOBKDM4EMEN1ALDH1A1
SCHEMBL5224566 0.84 MAPK14 (0.47) TAAR1MAOBHTR2CSLC6A4HTR2B
SCHEMBL1154474 0.83 CYP11B1 (0.43) MEN1ALDH1A1KMT2A
SCHEMBL5220371 0.82 HTR2C (0.44) TAAR1MAOBHTR2CSLC6A4HTR2B
SCHEMBL5217387 0.81 CASR (0.41) TAAR1MAOBMEN1ALDH1A1KMT2A
SCHEMBL5225071 0.81 CASR (0.51) SLC6A4
SCHEMBL5222695 0.80 MAPK14 (0.40) DRD2HTR2CSLC6A4HTR2BMEN1
SCHEMBL1154302 0.79 LMNA (0.43) TAAR1DRD2MAOBKMT2ATDP1
SCHEMBL5221531 0.79 CASR (0.41) TAAR1HTR1ASLC6A4
SCHEMBL22169493 0.77 RAB9A (0.47) MAOBKDM4EMEN1KMT2ASQOR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1765810-A1 2,4-DIAMINOQUINAZOLINES FOR SPINAL MUSCULAR ATROPHY Decode Chemistry, Inc. (US) 2007-03-28 EP disclosed
WO-2005123724-A1 2,4-DIAMINOQUINAZOLINES FOR SPINAL MUSCULAR ATROPHY DECODE CHEMISTRY, INC. (US) 2005-12-29 WO disclosed