SCHEMBL5220690

SCHEMBL5220690

N#Cc1cccnc1N1CCC(NC(=O)O)CC1

nearest known ligand 0.66

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 4/20 0.66
RECQL P46063 1/20 0.66
ACKR3 P25106 1/20 0.53
HSD11B1 P28845 2/20 0.53
MALT1 Q9UDY8 1/20 0.53
ALDH1A1 P00352 2/20 0.51
TDP1 Q9NUW8 1/20 0.51
HDAC2 Q92769 1/20 0.49
PANK3 Q9H999 1/20 0.49
CA12 O43570 1/20 0.48
CA1 P00915 1/20 0.48
CA2 P00918 1/20 0.48
CA9 Q16790 1/20 0.48
DRD2 P14416 1/20 0.48
HTR2A P28223 1/20 0.48
LDHA P00338 1/20 0.48
SSTR4 P31391 1/20 0.47
MAPT P10636 1/20 0.47
MEN1 O00255 1/20 0.47
CYP1A2 P05177 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3110161 0.83 KDM4E (0.79) KDM4ERECQLHSD11B1MALT1ALDH1A1
SCHEMBL27643840 0.83 KDM4E (0.57) KDM4ERECQLACKR3HSD11B1MALT1
SCHEMBL1727869 0.82 KDM4E (0.62) KDM4ERECQLACKR3HSD11B1MALT1
SCHEMBL1727561 0.81 KMT2A (0.48) KDM4ERECQLACKR3MALT1ALDH1A1
SCHEMBL5220685 0.81 MALT1 (0.64) MALT1MEN1CYP1A2CYP3A4CYP2C9
SCHEMBL1728915 0.81 KMT2A (0.50) KDM4ERECQLMALT1ALDH1A1MEN1
SCHEMBL31042527 0.80 DRD4 (0.51) KDM4EALDH1A1DRD2HTR2AMAPT
SCHEMBL1727887 0.80 KDM4E (0.60) KDM4ERECQLACKR3HSD11B1MALT1
SCHEMBL13622633 0.80 KDM4E (0.66) KDM4ERECQLACKR3HSD11B1MALT1
SCHEMBL3288507 0.80 KDM4E (0.51) KDM4ERECQLACKR3HSD11B1MALT1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1664025-B1 PYRROL DERIVATIVES WITH ANTIBACTERIAL ACTIVITY ASTRAZENECA AB (SE) 2007-09-19 EP disclosed