SCHEMBL5220920

SCHEMBL5220920

CCCCNC[C@H](O)[C@H](Cc1ccccc1)N(C(=O)O)C(C)(C)C

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
REN P00797 3/20 0.40
BCHE P06276 4/20 0.40
OPRM1 P35372 1/20 0.39
OPRD1 P41143 1/20 0.39
OPRK1 P41145 1/20 0.39
BACE1 P56817 3/20 0.39
CYP1A2 P05177 1/20 0.38
CYP2C9 P11712 1/20 0.38
CYP2C19 P33261 1/20 0.38
CTSK P43235 2/20 0.37
ANPEP P15144 1/20 0.37
ERAP2 Q6P179 1/20 0.37
CSNK1E P49674 1/20 0.37
CHRNB2 P17787 1/20 0.37
CHRNB4 P30926 1/20 0.37
CHRNA3 P32297 1/20 0.37
CHRNA4 P43681 1/20 0.37
CTSD P07339 1/20 0.37
ABCB1 P08183 2/20 0.37
HDAC3 O15379 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5220912 1.00 REN (0.40) RENBCHEOPRM1OPRD1OPRK1
SCHEMBL5223916 0.97 SIGMAR1 (0.41) RENBCHEOPRM1OPRD1OPRK1
SCHEMBL5223922 0.97 SIGMAR1 (0.41) RENBCHEOPRM1OPRD1OPRK1
SCHEMBL5224655 0.95 CSNK1E (0.41) BCHEOPRM1OPRD1OPRK1BACE1
SCHEMBL5224641 0.95 CSNK1E (0.41) BCHEOPRM1OPRD1OPRK1BACE1
SCHEMBL4516305 0.90 REN (0.51) RENHDAC3KDM4ETDP1
SCHEMBL4516309 0.90 REN (0.51) RENHDAC3KDM4ETDP1
SCHEMBL5219646 0.88 ADRB3 (0.43) BCHEOPRM1OPRD1OPRK1BACE1
SCHEMBL5219638 0.88 ADRB3 (0.43) BCHEOPRM1OPRD1OPRK1BACE1
SCHEMBL5218726 0.87 BCHE (0.42) BCHEOPRM1OPRD1OPRK1BACE1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1567488-B1 HYDROXYETHYLAMINE DERIVATIVES FOR THE TREATMENT OF ALZHEIMER'S DISEASE GLAXO GROUP LTD (GB) 2007-02-21 EP disclosed