SCHEMBL5221504

SCHEMBL5221504

CCc1c[nH]c2c(N3CCCC3=O)cc(C(=O)O)cc12

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CTSD P07339 1/20 0.51
BACE1 P56817 1/20 0.51
BACE2 Q9Y5Z0 1/20 0.51
ALDH1A1 P00352 2/20 0.41
CYP2C9 P11712 4/20 0.40
CYP3A4 P08684 2/20 0.40
HPGD P15428 2/20 0.40
CYP1A2 P05177 1/20 0.40
CYP2D6 P10635 1/20 0.40
CYP2C19 P33261 1/20 0.40
GAA P10253 1/20 0.37
PRKAB2 O43741 1/20 0.37
PRKAG1 P54619 1/20 0.37
PRKAA2 P54646 1/20 0.37
PRKAA1 Q13131 1/20 0.37
PRKAG3 Q9UGI9 1/20 0.37
PRKAG2 Q9UGJ0 1/20 0.37
PRKAB1 Q9Y478 1/20 0.37
HSD17B10 Q99714 1/20 0.36
USP2 O75604 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5221970 0.98 CTSD (0.49) CTSDBACE1BACE2ALDH1A1CYP2C9
SCHEMBL5222278 0.89 CTSD (0.48) CTSDBACE1BACE2ALDH1A1CYP2C9
SCHEMBL5221500 0.85 CTSD (0.46) CTSDBACE1BACE2ALDH1A1CYP3A4
SCHEMBL5219361 0.85 GAA (0.44) CTSDBACE1BACE2ALDH1A1CYP2C9
SCHEMBL5220565 0.83 CTSD (0.42) CTSDBACE1BACE2ALDH1A1CYP2C9
SCHEMBL5221844 0.78 HSD17B10 (0.43) CTSDBACE1BACE2ALDH1A1CYP2C9
SCHEMBL5390345 0.78 CTSD (0.42) CTSDBACE1BACE2ALDH1A1CYP2C9
SCHEMBL5222116 0.77 CASP1 (0.43) CTSDBACE1BACE2ALDH1A1MEN1
SCHEMBL5226004 0.77 CTSD (0.36) CTSDBACE1BACE2
SCHEMBL5226007 0.77 POLB (0.39) CTSDBACE1BACE2GAAF10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1567488-B1 HYDROXYETHYLAMINE DERIVATIVES FOR THE TREATMENT OF ALZHEIMER'S DISEASE GLAXO GROUP LTD (GB) 2007-02-21 EP disclosed