SCHEMBL5221531

SCHEMBL5221531

N#Cc1c(F)cccc1OCCc1ccc(Cl)c(Cl)c1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CASR P41180 5/20 0.41
NPC1 O15118 3/20 0.40
RAB9A P51151 3/20 0.40
PNMT P11086 1/20 0.40
TAAR1 Q96RJ0 1/20 0.40
MRGPRX4 Q96LA9 1/20 0.39
CYP2D6 P10635 2/20 0.37
CYP1A2 P05177 1/20 0.37
CYP2C9 P11712 1/20 0.37
CYP2C19 P33261 1/20 0.37
KCNH2 Q12809 3/20 0.37
SIGMAR1 Q99720 2/20 0.37
TMEM97 Q5BJF2 1/20 0.37
MAPT P10636 2/20 0.36
LMNA P02545 1/20 0.36
TSHR P16473 1/20 0.36
HTT P42858 1/20 0.36
GLA P06280 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
GPR84 Q9NQS5 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5220371 0.86 HTR2C (0.44) CASRNPC1RAB9ATAAR1MRGPRX4
SCHEMBL1155054 0.85 NPC1 (0.52) CASRNPC1RAB9ATAAR1MRGPRX4
SCHEMBL5217387 0.85 CASR (0.41) CASRNPC1RAB9ATAAR1KCNH2
SCHEMBL5224566 0.83 MAPK14 (0.47) CASRNPC1TAAR1MAPTLMNA
SCHEMBL5225071 0.82 CASR (0.51) CASRCYP2D6KCNH2MAPTLMNA
SCHEMBL5222695 0.81 MAPK14 (0.40) CASRNPC1RAB9AMRGPRX4MAPT
SCHEMBL1154474 0.81 CYP11B1 (0.43) NPC1RAB9AMRGPRX4MAPTLMNA
SCHEMBL1154302 0.80 LMNA (0.43) CASRNPC1RAB9ATAAR1CYP1A2
SCHEMBL1154219 0.79 NPC1 (0.51) CASRNPC1RAB9ATAAR1MRGPRX4
SCHEMBL5223526 0.79 HSD11B1 (0.43) CASRNPC1RAB9ATAAR1MRGPRX4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1765810-A1 2,4-DIAMINOQUINAZOLINES FOR SPINAL MUSCULAR ATROPHY Decode Chemistry, Inc. (US) 2007-03-28 EP disclosed
WO-2005123724-A1 2,4-DIAMINOQUINAZOLINES FOR SPINAL MUSCULAR ATROPHY DECODE CHEMISTRY, INC. (US) 2005-12-29 WO disclosed