SCHEMBL5221569

SCHEMBL5221569

CC(C)CC(C)NC[C@@H](O)[C@H](Cc1ccccc1)N(C(=O)O)C(C)(C)C

nearest known ligand 0.42

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 2/20 0.42
RAB9A P51151 2/20 0.42
ADRB2 P07550 4/20 0.40
ADRB1 P08588 1/20 0.40
ADRB3 P13945 1/20 0.40
TP53 P04637 1/20 0.39
CYP1A2 P05177 1/20 0.39
CYP2D6 P10635 1/20 0.39
ALOX15 P16050 1/20 0.39
TSHR P16473 1/20 0.39
CYP2C19 P33261 1/20 0.39
SIGMAR1 Q99720 1/20 0.39
PSMB5 P28074 1/20 0.38
MME P08473 1/20 0.38
LMNA P02545 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5221576 1.00 NPC1 (0.42) NPC1RAB9AADRB2ADRB1ADRB3
SCHEMBL5216511 0.89 TRPA1 (0.40) NPC1RAB9AADRB2ADRB1ADRB3
SCHEMBL5216515 0.89 TRPA1 (0.40) NPC1RAB9AADRB2ADRB1ADRB3
SCHEMBL609658 0.84 ANPEP (0.42) NPC1RAB9A
SCHEMBL609656 0.84 ANPEP (0.42) NPC1RAB9A
SCHEMBL5223473 0.83 OPRD1 (0.41) NPC1RAB9A
SCHEMBL5223463 0.83 OPRD1 (0.41) NPC1RAB9A
SCHEMBL5224996 0.81 OPRM1 (0.39) NPC1RAB9ACYP1A2CYP2C19
SCHEMBL5224985 0.81 OPRM1 (0.39) NPC1RAB9ACYP1A2CYP2C19
SCHEMBL4870053 0.80 ABCB1 (0.38) NPC1RAB9AADRB2ADRB1ADRB3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1567488-B1 HYDROXYETHYLAMINE DERIVATIVES FOR THE TREATMENT OF ALZHEIMER'S DISEASE GLAXO GROUP LTD (GB) 2007-02-21 EP disclosed