SCHEMBL5223460

SCHEMBL5223460

COc1cccc(CC(C)(C)NC[C@H](O)[C@H](Cc2ccccc2)N(C(=O)O)C(C)(C)C)c1

nearest known ligand 0.46

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
CASR P41180 4/20 0.46
CTSD P07339 11/20 0.46
ADRB2 P07550 1/20 0.43
ADRB1 P08588 1/20 0.43
BCHE P06276 1/20 0.43
MTNR1A P48039 1/20 0.43
MTNR1B P49286 1/20 0.43
BACE1 P56817 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5223457 1.00 CASR (0.46) CASRCTSDADRB2ADRB1BCHE
SCHEMBL5216401 0.87 OPRM1 (0.47) CTSDADRB2ADRB1BCHEBACE1
SCHEMBL5216394 0.87 OPRM1 (0.47) CTSDADRB2ADRB1BCHEBACE1
SCHEMBL5219027 0.86 CASR (0.41) CASRCTSDADRB2
SCHEMBL5219019 0.86 CASR (0.41) CASRCTSDADRB2
SCHEMBL5217991 0.83 CASR (0.41) CASRADRB2ADRB1BACE1
SCHEMBL5224863 0.82 KDM4E (0.43) CTSDADRB2ADRB1BCHEBACE1
SCHEMBL5224856 0.82 KDM4E (0.43) CTSDADRB2ADRB1BCHEBACE1
SCHEMBL5223492 0.82 OPRM1 (0.40) CASRADRB2ADRB1BCHEBACE1
SCHEMBL5223500 0.82 OPRM1 (0.40) CASRADRB2ADRB1BCHEBACE1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1567488-B1 HYDROXYETHYLAMINE DERIVATIVES FOR THE TREATMENT OF ALZHEIMER'S DISEASE GLAXO GROUP LTD (GB) 2007-02-21 EP disclosed