SCHEMBL5224073

SCHEMBL5224073

COc1ccc2c(c1)C(NC[C@@H](O)[C@H](Cc1ccccc1)N(C(=O)O)C(C)(C)C)CC2

nearest known ligand 0.48

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 3/20 0.48
CTSD P07339 2/20 0.48
BACE2 Q9Y5Z0 1/20 0.48
ACHE P22303 8/20 0.46
KDM1A O60341 2/20 0.42
MAOA P21397 2/20 0.42
MAOB P27338 2/20 0.42
GRIN1 Q05586 1/20 0.39
GRIN2B Q13224 1/20 0.39
MTNR1A P48039 4/20 0.39
XIAP P98170 1/20 0.39
MTNR1B P49286 3/20 0.39
NQO2 P16083 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5224081 1.00 BACE1 (0.48) BACE1CTSDBACE2ACHEKDM1A
SCHEMBL5218168 0.87 CTSD (0.44) BACE1CTSDBACE2ACHEMAOA
SCHEMBL5218164 0.87 CTSD (0.44) BACE1CTSDBACE2ACHEMAOA
SCHEMBL5223365 0.81 CTSD (0.49) BACE1CTSDBACE2ACHEKDM1A
SCHEMBL7613311 0.76 BACE1 (0.60) BACE1CTSDBACE2KDM1AMAOA
SCHEMBL7613304 0.76 BACE1 (0.60) BACE1CTSDBACE2KDM1AMAOA
SCHEMBL4045255 0.75 KDM1A (0.49) BACE1CTSDBACE2KDM1AMAOA
SCHEMBL4041567 0.75 KDM1A (0.49) BACE1CTSDBACE2KDM1AMAOA
SCHEMBL5223460 0.74 CASR (0.46) BACE1CTSDMTNR1AMTNR1B
SCHEMBL5223457 0.74 CASR (0.46) BACE1CTSDMTNR1AMTNR1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1567488-B1 HYDROXYETHYLAMINE DERIVATIVES FOR THE TREATMENT OF ALZHEIMER'S DISEASE GLAXO GROUP LTD (GB) 2007-02-21 EP disclosed