SCHEMBL5224286

SCHEMBL5224286

O=C(O)NC1CCN(c2cc(C(=O)NCCCN3CCOCC3)cc(Cl)n2)CC1

nearest known ligand 0.52

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
MAPK14 Q16539 1/20 0.51
KDM4E B2RXH2 1/20 0.49
ALDH1A1 P00352 1/20 0.49
SMN1; SMN2 Q16637 1/20 0.49
KMT2A Q03164 2/20 0.47
TSHR P16473 1/20 0.47
MEN1 O00255 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5220732 0.95 HPGDS (0.50) KDM4EALDH1A1
SCHEMBL3289122 0.87 MAPK14 (0.47) MAPK14KMT2AMEN1
Hydrochloric Acid SCHEMBL3282645 0.87 SMN1; SMN2 (0.49) KDM4EALDH1A1SMN1; SMN2KMT2ATSHR
SCHEMBL3285361 0.86 MAPK14 (0.46) MAPK14KMT2ATSHRMEN1
SCHEMBL3281794 0.83 HPGDS (0.45)
Hydrochloric Acid SCHEMBL3280894 0.82 ALDH1A1 (0.51) KDM4EALDH1A1TSHR
SCHEMBL5222020 0.82 SMN1; SMN2 (0.67) KDM4EALDH1A1SMN1; SMN2TSHR
SCHEMBL3282345 0.82 HPGDS (0.45) MAPK14KDM4EALDH1A1
SCHEMBL3281618 0.80 LMNA (0.45) ALDH1A1SMN1; SMN2KMT2ATSHRMEN1
SCHEMBL23608032 0.79 KDM4E (0.47) KDM4ESMN1; SMN2KMT2AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1664025-B1 PYRROL DERIVATIVES WITH ANTIBACTERIAL ACTIVITY ASTRAZENECA AB (SE) 2007-09-19 EP disclosed