SCHEMBL5225473

SCHEMBL5225473

COc1ccc2sc(OC(=O)Nc3nnn[nH]3)c(SCC3CCCCC3)c2c1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
METAP2 P50579 3/20 0.38
CYP1A2 P05177 1/20 0.37
CYP2E1 P05181 1/20 0.37
CYP3A4 P08684 1/20 0.37
CYP2C8 P10632 1/20 0.37
CYP2D6 P10635 1/20 0.37
CYP2C9 P11712 1/20 0.37
CYP2B6 P20813 1/20 0.37
CYP2C19 P33261 1/20 0.37
USP2 O75604 1/20 0.36
ALDH1A1 P00352 1/20 0.36
LMNA P02545 1/20 0.36
NPSR1 Q6W5P4 1/20 0.36
MAOA P21397 1/20 0.35
MAOB P27338 1/20 0.35
NPC1 O15118 3/20 0.34
RAB9A P51151 3/20 0.34
GCK P35557 1/20 0.34
MAPT P10636 2/20 0.34
MPO P05164 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5225831 0.89 METAP2 (0.37) METAP2ALDH1A1NPSR1NPC1RAB9A
SCHEMBL5227538 0.88 MPO (0.36) CYP1A2CYP3A4CYP2C9CYP2C19USP2
SCHEMBL5224808 0.87 MPO (0.37) USP2ALDH1A1LMNANPSR1MAOA
SCHEMBL5225302 0.76 PIK3CD (0.32)
SCHEMBL5226252 0.75 PIK3CD (0.32) ALDH1A1MAPT
SCHEMBL4766147 0.74 EDNRA (0.45) CYP1A2CYP2E1CYP3A4CYP2C8CYP2D6
SCHEMBL5228680 0.74 PIK3CD (0.38)
SCHEMBL5226593 0.73 PIK3CD (0.31)
SCHEMBL5227163 0.73 POLB (0.31) KMT2A
SCHEMBL5767040 0.72 PIK3CD (0.39) METAP2NPC1RAB9AMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1636212-B1 CYCLOALKYLSULFANYL SUBSTITUTED BENZO¬B|THIOPHENES AS THERAPEUTIC AGENTS WARNER LAMBERT CO (US) 2007-06-27 EP claimed