SCHEMBL5226460

SCHEMBL5226460

OC1CCN(C(c2ccc(-c3ccc4c(c3)OCO4)cc2)c2cn[nH]c2-c2ccco2)C1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.38
KDM4E B2RXH2 3/20 0.38
GAA P10253 3/20 0.38
POLB P06746 2/20 0.38
HPGD P15428 2/20 0.38
ALOX15 P16050 2/20 0.38
TSHR P16473 2/20 0.38
SMN1; SMN2 Q16637 2/20 0.38
HSD17B10 Q99714 2/20 0.38
NPC1 O15118 1/20 0.38
TP53 P04637 1/20 0.38
PKM P14618 1/20 0.38
RAB9A P51151 1/20 0.38
NPSR1 Q6W5P4 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.36
KDM4D Q6B0I6 5/20 0.36
KMT2A Q03164 4/20 0.35
MEN1 O00255 3/20 0.35
ADORA3 P0DMS8 1/20 0.35
ADORA2A P29274 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5227650 0.95 SIRT1 (0.35) ALDH1A1KDM4EGAAPOLBHPGD
SCHEMBL5228511 0.84 MAPT (0.38) ALDH1A1KDM4EPOLBHPGDTSHR
SCHEMBL2003026 0.80 GSK3B (0.33) ALDH1A1GAAMAPTLMNA
SCHEMBL1998839 0.80 GSK3B (0.34) ALDH1A1GAAKDM4DLMNA
SCHEMBL1998346 0.79 GSK3B (0.34) SMN1; SMN2NPC1RAB9AL3MBTL1MAPT
SCHEMBL2001021 0.79 LMNA (0.33) ALDH1A1GAAADORA2AMAPTLMNA
SCHEMBL2000118 0.79 KCNH2 (0.33) ALDH1A1GAASMN1; SMN2NPC1RAB9A
SCHEMBL2908342 0.78 ITGB2 (0.38) ALDH1A1KDM4EGAAPOLBHPGD
SCHEMBL5907357 0.71 HTR1A (0.39) ALDH1A1KMT2ALMNA
SCHEMBL5228031 0.70 MAPK1 (0.40) MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1611122-B1 SUBSTITUTED PYRAZOLE COMPOUNDS MERCK PATENT GMBH (DE) 2007-06-13 EP disclosed