SCHEMBL5227650

SCHEMBL5227650

OC1CCN(C(c2ccc(-c3ccc4c(c3)OCCO4)cc2)c2cn[nH]c2-c2ccco2)C1

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SIRT1 Q96EB6 1/20 0.35
ITGB2 P05107 2/20 0.35
ICAM1 P05362 2/20 0.35
ITGAL P20701 2/20 0.35
ALDH1A1 P00352 5/20 0.34
ALOX15 P16050 2/20 0.34
LMNA P02545 2/20 0.34
ALOX12 P18054 1/20 0.34
HTT P42858 1/20 0.34
CLK1 P49759 1/20 0.34
FAAH O00519 1/20 0.33
KCNH2 Q12809 1/20 0.33
PTK2 Q05397 1/20 0.33
HSP90AA1 P07900 1/20 0.33
POLB P06746 3/20 0.32
KDM4E B2RXH2 1/20 0.32
NPC1 O15118 1/20 0.32
TP53 P04637 1/20 0.32
GAA P10253 1/20 0.32
PKM P14618 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5226460 0.95 ALDH1A1 (0.38) SIRT1ALDH1A1ALOX15LMNAALOX12
SCHEMBL5228511 0.84 MAPT (0.38) ALDH1A1HTTPOLBKDM4ENPC1
SCHEMBL2908342 0.83 ITGB2 (0.38) SIRT1ITGB2ICAM1ITGALALDH1A1
SCHEMBL1998839 0.80 GSK3B (0.34) ALDH1A1LMNAGAAKDM4D
SCHEMBL2003026 0.80 GSK3B (0.33) ALDH1A1LMNAGAA
SCHEMBL1998346 0.79 GSK3B (0.34) ITGB2ICAM1ITGALLMNANPC1
SCHEMBL2001021 0.79 LMNA (0.33) ALDH1A1LMNAKCNH2GAA
SCHEMBL2000118 0.79 KCNH2 (0.33) ALDH1A1LMNAKCNH2NPC1GAA
SCHEMBL5907357 0.71 HTR1A (0.39) ALDH1A1LMNAKMT2A
SCHEMBL5907259 0.70 P4HB (0.40) ALDH1A1ALOX15LMNAALOX12HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1611122-B1 SUBSTITUTED PYRAZOLE COMPOUNDS MERCK PATENT GMBH (DE) 2007-06-13 EP disclosed