SCHEMBL5226495

SCHEMBL5226495

COc1ccc(-c2ccc(C(c3cn[nH]c3-c3ccco3)N3CCN(C4CCCC4)CC3)cc2)cc1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPSR1 Q6W5P4 5/20 0.44
ALDH1A1 P00352 4/20 0.44
MEN1 O00255 2/20 0.44
KMT2A Q03164 2/20 0.44
KDM4E B2RXH2 1/20 0.44
HTT P42858 1/20 0.44
TSHR P16473 3/20 0.43
LMNA P02545 2/20 0.42
NPC1 O15118 1/20 0.42
TAAR1 Q96RJ0 1/20 0.42
CHRM2 P08172 10/20 0.42
CHRM1 P11229 10/20 0.42
CHRM4 P08173 5/20 0.41
CHRM3 P20309 4/20 0.41
USP2 O75604 1/20 0.41
CHRM5 P08912 2/20 0.39
CCR3 P51677 1/20 0.39
MAPT P10636 1/20 0.39
RXFP1 Q9HBX9 1/20 0.38
HRH3 Q9Y5N1 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2761178 0.89 TSHR (0.48) NPSR1ALDH1A1MEN1KMT2AHTT
SCHEMBL5232268 0.87 BCL2L11 (0.39) ALDH1A1MEN1KMT2AKDM4EHTT
SCHEMBL5224311 0.86 LMNA (0.45) ALDH1A1MEN1KMT2AHTTTSHR
SCHEMBL5230462 0.86 HTR1A (0.47) ALDH1A1MEN1KMT2AKDM4EHTT
SCHEMBL5228511 0.83 MAPT (0.38) ALDH1A1MEN1KMT2AKDM4EHTT
SCHEMBL2761079 0.79 TSHR (0.40) NPSR1ALDH1A1MEN1KMT2AHTT
SCHEMBL2761138 0.76 LMNA (0.40) NPSR1HTTLMNAUSP2MAPT
SCHEMBL2761010 0.76 MAPT (0.41) NPSR1HTTLMNACHRM2CHRM1
SCHEMBL2761238 0.75 LMNA (0.51) NPSR1ALDH1A1MEN1KMT2AKDM4E
Hydrochloric Acid SCHEMBL1997591 0.74 LMNA (0.50) NPSR1ALDH1A1MEN1KMT2AKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1611122-B1 SUBSTITUTED PYRAZOLE COMPOUNDS MERCK PATENT GMBH (DE) 2007-06-13 EP disclosed