SCHEMBL5226715

SCHEMBL5226715

CC(C)(C)OC(=O)ON1CCN(Cc2cnn(-c3ccc(-c4ccc5c(c4)OCO5)cc3)c2-c2ccco2)CC1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 7/20 0.37
TP53 P04637 5/20 0.37
LMNA P02545 3/20 0.37
USP2 O75604 2/20 0.37
SMN1; SMN2 Q16637 2/20 0.37
SCD5 Q86SK9 1/20 0.37
THRB P10828 1/20 0.36
PKM P14618 2/20 0.36
FABP1 P07148 1/20 0.36
FABP6 P51161 1/20 0.36
MAPT P10636 3/20 0.36
POLB P06746 4/20 0.35
KDM4E B2RXH2 3/20 0.35
TSHR P16473 2/20 0.35
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35
NPC1 O15118 2/20 0.34
RAB9A P51151 2/20 0.34
GAA P10253 1/20 0.34
HPGD P15428 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5224994 0.96 MAPT (0.35) ALDH1A1TP53LMNAUSP2SMN1; SMN2
SCHEMBL5226151 0.88 SMO (0.35) ALDH1A1TP53LMNAUSP2KDM4E
SCHEMBL5224989 0.86 SCD5 (0.44) TP53LMNASCD5THRBMAPT
SCHEMBL5222920 0.83 ALDH1A1 (0.41) ALDH1A1TP53LMNAUSP2SMN1; SMN2
SCHEMBL5226166 0.83 ALDH1A1 (0.41) ALDH1A1TP53LMNAUSP2SMN1; SMN2
SCHEMBL5225926 0.81 MCHR1 (0.41) ALDH1A1TP53LMNAUSP2SMN1; SMN2
SCHEMBL5226838 0.80 ALDH1A1 (0.41) ALDH1A1TP53LMNAUSP2SMN1; SMN2
SCHEMBL5230509 0.79 POLB (0.41) ALDH1A1TP53SMN1; SMN2PKMPOLB
SCHEMBL5229195 0.79 POLB (0.40) ALDH1A1TP53LMNAUSP2SMN1; SMN2
SCHEMBL5229335 0.78 ALDH1A1 (0.42) ALDH1A1TP53LMNAUSP2SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1611122-B1 SUBSTITUTED PYRAZOLE COMPOUNDS MERCK PATENT GMBH (DE) 2007-06-13 EP disclosed