SCHEMBL5226838

SCHEMBL5226838

c1coc(-c2c(CN3CCNCC3)cnn2-c2ccc(-c3ccc4c(c3)OCO4)cc2)c1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.41
ALOX15 P16050 2/20 0.41
TP53 P04637 2/20 0.41
SMN1; SMN2 Q16637 2/20 0.41
GAA P10253 2/20 0.41
KDM4E B2RXH2 1/20 0.41
NPC1 O15118 1/20 0.41
POLB P06746 1/20 0.41
PKM P14618 1/20 0.41
HPGD P15428 1/20 0.41
TSHR P16473 1/20 0.41
RAB9A P51151 1/20 0.41
NPSR1 Q6W5P4 1/20 0.41
HSD17B10 Q99714 1/20 0.41
CHRM3 P20309 9/20 0.38
CHRM1 P11229 1/20 0.38
PDCD1 Q15116 1/20 0.38
CD274 Q9NZQ7 1/20 0.38
CYP1A2 P05177 2/20 0.38
CYP3A4 P08684 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5227547 0.95 PDCD1 (0.43) ALDH1A1ALOX15TP53SMN1; SMN2GAA
SCHEMBL5230401 0.90 ALDH1A1 (0.38) ALDH1A1ALOX15TP53SMN1; SMN2GAA
SCHEMBL5222920 0.89 ALDH1A1 (0.41) ALDH1A1ALOX15TP53SMN1; SMN2GAA
SCHEMBL5226166 0.89 ALDH1A1 (0.41) ALDH1A1ALOX15TP53SMN1; SMN2GAA
SCHEMBL5229335 0.87 ALDH1A1 (0.42) ALDH1A1ALOX15TP53SMN1; SMN2GAA
SCHEMBL5224744 0.85 HTR1A (0.38) ALDH1A1KDM4EHPGDTSHRCHRM3
SCHEMBL5226663 0.85 KMT2A (0.44) ALDH1A1ALOX15TP53SMN1; SMN2GAA
SCHEMBL5229195 0.84 POLB (0.40) ALDH1A1ALOX15TP53SMN1; SMN2GAA
SCHEMBL5230509 0.84 POLB (0.41) ALDH1A1ALOX15TP53SMN1; SMN2GAA
SCHEMBL5226446 0.84 ALDH1A1 (0.41) ALDH1A1ALOX15TP53SMN1; SMN2GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1611122-B1 SUBSTITUTED PYRAZOLE COMPOUNDS MERCK PATENT GMBH (DE) 2007-06-13 EP disclosed