SCHEMBL5226745

SCHEMBL5226745

CN1CCN(Cc2cnn(-c3ccc(C4=C(Cc5ccccc5)OCO4)cc3)c2-c2ccccc2F)CC1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMO Q99835 5/20 0.38
DRD4 P21917 3/20 0.38
DRD3 P35462 2/20 0.38
DRD2 P14416 1/20 0.38
SSTR5 P35346 1/20 0.37
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35
MAPK14 Q16539 1/20 0.34
MC4R P32245 1/20 0.34
ALDH1A1 P00352 1/20 0.34
MAP4K1 Q92918 1/20 0.34
ACHE P22303 1/20 0.34
JAK2 O60674 1/20 0.33
JAK1 P23458 1/20 0.33
TYK2 P29597 1/20 0.33
JAK3 P52333 1/20 0.33
ADORA2A P29274 1/20 0.33
ADORA1 P30542 1/20 0.33
MAPK1 P28482 1/20 0.33
STAT1 P42224 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5222928 0.85 SMO (0.38) SMODRD4DRD3DRD2MEN1
SCHEMBL1689504 0.84 SMO (0.45) SMODRD4DRD3DRD2SSTR5
SCHEMBL7256544 0.83 DRD4 (0.44) SMODRD4DRD3DRD2SSTR5
SCHEMBL5737789 0.82 SMO (0.44) SMODRD4DRD3DRD2SSTR5
SCHEMBL7261049 0.81 CHKA (0.50) SMODRD4DRD3DRD2SSTR5
SCHEMBL2761054 0.81 MAPT (0.43) DRD4DRD3SSTR5ALDH1A1MAPK1
SCHEMBL5228638 0.80 DRD4 (0.41) SMODRD4DRD3DRD2SSTR5
SCHEMBL5227102 0.80 LMNA (0.44) SMODRD4DRD3DRD2SSTR5
SCHEMBL5225912 0.79 MAP4K1 (0.41) SMODRD4DRD3DRD2SSTR5
SCHEMBL5224217 0.79 SMO (0.44) SMODRD4DRD3DRD2SSTR5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1611122-B1 SUBSTITUTED PYRAZOLE COMPOUNDS MERCK PATENT GMBH (DE) 2007-06-13 EP disclosed