SCHEMBL5222928

SCHEMBL5222928

CN1CCN(Cc2cnn(-c3ccc(C4=C(Cc5ccccc5)OCO4)cc3)c2-c2ccco2)CC1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMO Q99835 3/20 0.38
DRD4 P21917 3/20 0.38
DRD3 P35462 3/20 0.38
DRD2 P14416 2/20 0.38
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35
HCRTR1 O43613 1/20 0.34
MC4R P32245 1/20 0.34
L3MBTL1 Q9Y468 3/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
ALDH1A1 P00352 4/20 0.33
MAPT P10636 3/20 0.33
KDM4E B2RXH2 2/20 0.33
NPSR1 Q6W5P4 1/20 0.33
TDP1 Q9NUW8 1/20 0.33
TP53 P04637 1/20 0.33
POLB P06746 1/20 0.33
CHKA P35790 1/20 0.32
KDM5B Q9UGL1 2/20 0.32
ALK Q9UM73 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5226173 0.93 SMO (0.38) SMODRD4DRD3DRD2MEN1
SCHEMBL5226844 0.90 SIGMAR1 (0.34) SMODRD4DRD3DRD2MEN1
SCHEMBL5229345 0.88 EGFR (0.34) SMODRD4DRD3DRD2MEN1
SCHEMBL5226667 0.88 DRD4 (0.39) SMODRD4DRD3DRD2MEN1
SCHEMBL5226450 0.85 F10 (0.35) KMT2AALDH1A1
SCHEMBL5226745 0.85 SMO (0.38) SMODRD4DRD3DRD2MEN1
SCHEMBL5229304 0.84 ALDH1A1 (0.33) SMN1; SMN2ALDH1A1MAPTKDM4ENPSR1
SCHEMBL5230408 0.84 SLC2A1 (0.32) HCRTR1L3MBTL1SMN1; SMN2ALDH1A1MAPT
SCHEMBL5225471 0.84 HRH3 (0.35) SMODRD4DRD3DRD2KDM4E
SCHEMBL5224860 0.83 ALDH1A1 (0.31) ALDH1A1MAPTKDM4ELMNAHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1611122-B1 SUBSTITUTED PYRAZOLE COMPOUNDS MERCK PATENT GMBH (DE) 2007-06-13 EP disclosed