SCHEMBL5226784

SCHEMBL5226784

COC(=O)c1cc(Br)cc(N2CCCS2(=O)=O)c1F

nearest known ligand 0.39

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
PIK3C3 Q8NEB9 2/20 0.39
TP53 P04637 4/20 0.36
OPRK1 P41145 9/20 0.35
CTSD P07339 1/20 0.34
BACE1 P56817 1/20 0.34
BACE2 Q9Y5Z0 1/20 0.34
SOS1 Q07889 1/20 0.34
KDM4E B2RXH2 1/20 0.34
NPC1 O15118 1/20 0.34
RAB9A P51151 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
NPSR1 Q6W5P4 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5217755 0.96 CTSD (0.37) PIK3C3OPRK1CTSDBACE1BACE2
SCHEMBL5226788 0.88 OPRK1 (0.35) OPRK1SOS1
SCHEMBL5223775 0.85 KDM4E (0.39) PIK3C3TP53OPRK1CTSDBACE1
SCHEMBL2366209 0.82 NR4A2 (0.42) PIK3C3TP53KDM4ENPC1RAB9A
SCHEMBL5224667 0.82 PIK3C3 (0.37) PIK3C3TP53CTSDBACE1BACE2
SCHEMBL5224665 0.82 PIK3C3 (0.37) PIK3C3TP53CTSDBACE1BACE2
SCHEMBL5223229 0.82 KDM4E (0.41) PIK3C3TP53OPRK1CTSDBACE1
SCHEMBL5221011 0.81 CTSD (0.39) PIK3C3TP53CTSDBACE1BACE2
SCHEMBL5221774 0.81 BACE1 (0.49) PIK3C3TP53CTSDBACE1BACE2
SCHEMBL5218540 0.81 ALDH1A1 (0.43) PIK3C3OPRK1KDM4ENPC1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1567488-B1 HYDROXYETHYLAMINE DERIVATIVES FOR THE TREATMENT OF ALZHEIMER'S DISEASE GLAXO GROUP LTD (GB) 2007-02-21 EP disclosed