SCHEMBL5224744

SCHEMBL5224744

Fc1cccc(-c2ccc(-n3ncc(CN4CCNCC4)c3-c3ccco3)cc2)c1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 3/20 0.38
HTR7 P34969 3/20 0.38
HTR1D P28221 2/20 0.38
HTR2A P28223 2/20 0.38
HTR2B P41595 2/20 0.38
HTR6 P50406 2/20 0.38
HTR1B P28222 1/20 0.38
HTR2C P28335 1/20 0.38
CHRM3 P20309 1/20 0.36
SMO Q99835 2/20 0.36
DHODH Q02127 1/20 0.36
HTR3A P46098 1/20 0.36
MEN1 O00255 2/20 0.35
KMT2A Q03164 2/20 0.35
NR1H2 P55055 1/20 0.35
BCL2A1 Q16548 1/20 0.35
KISS1R Q969F8 1/20 0.34
ALDH1A1 P00352 2/20 0.34
KDM4E B2RXH2 1/20 0.34
LMNA P02545 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5228536 0.90 EGFR (0.38) HTR6DHODHMEN1KMT2AALDH1A1
SCHEMBL5226613 0.89 SMO (0.40) SMODHODHMEN1KMT2AKISS1R
SCHEMBL5224673 0.89 SMO (0.40) HTR6SMODHODHKISS1RALDH1A1
SCHEMBL5229287 0.87 EGFR (0.40) SMODHODHMEN1KMT2AALDH1A1
SCHEMBL5226838 0.85 ALDH1A1 (0.41) CHRM3MEN1KMT2AALDH1A1KDM4E
SCHEMBL5226986 0.85 DRD4 (0.39) SMOALDH1A1KDM4ELMNAALPL
SCHEMBL5227547 0.84 PDCD1 (0.43) CHRM3ALDH1A1KDM4ELMNAACVR1
SCHEMBL5228047 0.84 HTR2C (0.37) HTR2CDHODHALDH1A1KDM4EROCK2
SCHEMBL2004259 0.83 HTR1A (0.35) HTR1AHTR7HTR2BHTR6SMO
SCHEMBL5230456 0.83 SMO (0.46) HTR1AHTR7HTR2BHTR6HTR1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1611122-B1 SUBSTITUTED PYRAZOLE COMPOUNDS MERCK PATENT GMBH (DE) 2007-06-13 EP disclosed