SCHEMBL5227547

SCHEMBL5227547

c1coc(-c2c(CN3CCNCC3)cnn2-c2ccc(-c3ccc4c(c3)OCCO4)cc2)c1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDCD1 Q15116 2/20 0.43
CD274 Q9NZQ7 2/20 0.43
TGFBR1 P36897 1/20 0.41
ACVR1 Q04771 1/20 0.41
CCND1 P24385 2/20 0.38
CDK6 Q00534 2/20 0.38
ALDH1A1 P00352 5/20 0.37
PKM P14618 2/20 0.37
HPGD P15428 2/20 0.37
SIRT1 Q96EB6 1/20 0.37
POLB P06746 2/20 0.36
TP53 P04637 2/20 0.36
SMN1; SMN2 Q16637 2/20 0.36
ALOX15 P16050 2/20 0.36
KDM4E B2RXH2 1/20 0.36
NPC1 O15118 1/20 0.36
GAA P10253 1/20 0.36
TSHR P16473 1/20 0.36
RAB9A P51151 1/20 0.36
NPSR1 Q6W5P4 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5226838 0.95 ALDH1A1 (0.41) PDCD1CD274TGFBR1ACVR1ALDH1A1
SCHEMBL5229195 0.89 POLB (0.40) PDCD1CD274CCND1CDK6ALDH1A1
SCHEMBL5230509 0.89 POLB (0.41) PDCD1CD274CCND1CDK6ALDH1A1
SCHEMBL5226174 0.88 ALDH1A1 (0.38) PDCD1CD274TGFBR1ACVR1ALDH1A1
SCHEMBL5225260 0.85 KMT2A (0.39) PDCD1CD274ALDH1A1PKMHPGD
SCHEMBL5230401 0.85 ALDH1A1 (0.38) PDCD1CD274ALDH1A1PKMHPGD
SCHEMBL5222920 0.84 ALDH1A1 (0.41) ALDH1A1PKMHPGDSIRT1POLB
SCHEMBL5226166 0.84 ALDH1A1 (0.41) CCND1CDK6ALDH1A1PKMHPGD
SCHEMBL5224744 0.84 HTR1A (0.38) ACVR1ALDH1A1HPGDKDM4ETSHR
SCHEMBL5227634 0.84 PDCD1 (0.40) PDCD1CD274ALDH1A1PKMHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1611122-B1 SUBSTITUTED PYRAZOLE COMPOUNDS MERCK PATENT GMBH (DE) 2007-06-13 EP disclosed