SCHEMBL5228410

SCHEMBL5228410

COc1ccc(-c2ccc(-n3ncc(CN)c3-c3ccco3)cc2)cc1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS1 P23219 1/20 0.49
PTGS2 P35354 1/20 0.49
NPBWR1 P48145 2/20 0.48
MCHR1 Q99705 1/20 0.48
TP53 P04637 4/20 0.45
KDM4E B2RXH2 4/20 0.45
MAPT P10636 2/20 0.43
HPGD P15428 2/20 0.41
HSD17B10 Q99714 2/20 0.41
ALDH1A1 P00352 2/20 0.41
TSHR P16473 1/20 0.41
HIF1A Q16665 1/20 0.41
SMN1; SMN2 Q16637 2/20 0.41
NPC1 O15118 1/20 0.41
RAB9A P51151 1/20 0.41
NPSR1 Q6W5P4 2/20 0.41
ADORA2A P29274 2/20 0.40
HTT P42858 2/20 0.40
LMNA P02545 1/20 0.40
GAA P10253 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5226619 0.87 NPBWR1 (0.47) PTGS1PTGS2NPBWR1MCHR1TP53
SCHEMBL5224717 0.85 NPBWR1 (0.45) PTGS1PTGS2NPBWR1MCHR1TP53
SCHEMBL5224302 0.82 SMO (0.49) PTGS1PTGS2NPBWR1MCHR1TP53
SCHEMBL5232263 0.82 SMO (0.49) PTGS1PTGS2NPBWR1MCHR1TP53
SCHEMBL5225666 0.81 NPBWR1 (0.43) PTGS1PTGS2NPBWR1MCHR1TP53
SCHEMBL5230456 0.81 SMO (0.46) PTGS1PTGS2NPBWR1MCHR1TP53
SCHEMBL5230220 0.81 NPBWR1 (0.40) PTGS1PTGS2NPBWR1MCHR1TP53
SCHEMBL5230237 0.79 MAPT (0.47) PTGS1PTGS2NPBWR1MCHR1TP53
SCHEMBL5228505 0.79 F10 (0.48)
SCHEMBL5226484 0.78 SMO (0.45) PTGS1PTGS2NPBWR1MCHR1TP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1611122-B1 SUBSTITUTED PYRAZOLE COMPOUNDS MERCK PATENT GMBH (DE) 2007-06-13 EP disclosed