SCHEMBL5228717

SCHEMBL5228717

COc1cccc(-c2c(C3CCCCC3)c3sc(OC(=O)O)cc3n2CC(=O)N(C)C)c1

nearest known ligand 0.63

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.38
HTT P42858 1/20 0.38
HIF1A Q16665 1/20 0.38
TSPO P30536 1/20 0.37
CYP2D6 P10635 1/20 0.37
HRH1 P35367 1/20 0.37
KCNH2 Q12809 1/20 0.37
JAK2 O60674 1/20 0.37
JAK3 P52333 1/20 0.37
PTK2 Q05397 1/20 0.37
ABL1 P00519 1/20 0.36
EGFR P00533 1/20 0.36
SRC P12931 1/20 0.36
ABL2 P42684 1/20 0.36
OPRK1 P41145 1/20 0.36
TP53 P04637 2/20 0.35
MAPT P10636 2/20 0.35
LMNA P02545 1/20 0.35
MEN1 O00255 2/20 0.35
KMT2A Q03164 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5233817 0.91 CYP2D6 (0.38) ALDH1A1CYP2D6HRH1KCNH2MAPT
SCHEMBL5231037 0.90 GRIN2B (0.38) TSPOCYP2D6HRH1KCNH2OPRK1
SCHEMBL2996782 0.89 ALDH1A1 (0.39) ALDH1A1HTTHIF1ATSPOCYP2D6
SCHEMBL5227499 0.89 TSPO (0.34) TSPOCYP2D6HRH1KCNH2EGFR
SCHEMBL5229499 0.89 CYP2D6 (0.34) CYP2D6HRH1KCNH2MAPT
SCHEMBL5232300 0.85 CYP2D6 (0.33) TSPOCYP2D6HRH1KCNH2MAPT
SCHEMBL5231299 0.84 CYP2D6 (0.33) CYP2D6HRH1KCNH2MAPT
SCHEMBL5231760 0.84 SCN9A (0.37) CYP2D6HRH1KCNH2MAPT
SCHEMBL5229100 0.84 PDE5A (0.39) CYP2D6HRH1KCNH2
SCHEMBL5233042 0.83 CYP2D6 (0.39) ALDH1A1CYP2D6HRH1KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1664059-B1 THIENOPYRROLES AS ANTIVIRAL AGENTS ANGELETTI P IST RICHERCHE BIO (IT) 2007-09-12 EP claimed