SCHEMBL5229100

SCHEMBL5229100

COc1ccc(-c2c(C3CCCCC3)c3sc(OC(=O)O)cc3n2CC(=O)N(C)C)cn1

nearest known ligand 0.57

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
PDE5A O76074 2/20 0.39
GRIN2B Q13224 7/20 0.38
GRIN1 Q05586 5/20 0.38
CYP3A4 P08684 1/20 0.36
CYP2C19 P33261 1/20 0.36
FYN P06241 1/20 0.36
ALOX5AP P20292 1/20 0.36
SCD O00767 1/20 0.35
SCD5 Q86SK9 1/20 0.35
CYP2D6 P10635 1/20 0.34
HRH1 P35367 1/20 0.34
KCNH2 Q12809 1/20 0.34
CPT2 P23786 1/20 0.34
CPT1A P50416 1/20 0.34
PIK3CA P42336 2/20 0.34
MTOR P42345 2/20 0.34
PDE6A P16499 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3000679 0.89 PDE5A (0.39) PDE5AGRIN2BGRIN1CYP3A4CYP2C19
SCHEMBL5233817 0.86 CYP2D6 (0.38) GRIN2BGRIN1CYP2D6HRH1KCNH2
SCHEMBL5232300 0.86 CYP2D6 (0.33) GRIN2BGRIN1CYP2D6HRH1KCNH2
SCHEMBL5231299 0.84 CYP2D6 (0.33) GRIN2BGRIN1CYP2D6HRH1KCNH2
SCHEMBL5228717 0.84 ALDH1A1 (0.38) CYP2D6HRH1KCNH2
SCHEMBL5233042 0.83 CYP2D6 (0.39) GRIN2BGRIN1CYP2D6HRH1KCNH2
SCHEMBL5231760 0.83 SCN9A (0.37) GRIN2BGRIN1CYP3A4CYP2C19CYP2D6
SCHEMBL5231037 0.82 GRIN2B (0.38) GRIN2BGRIN1CYP2D6HRH1KCNH2
SCHEMBL5227499 0.81 TSPO (0.34) GRIN2BGRIN1CYP2D6HRH1KCNH2
SCHEMBL5229499 0.81 CYP2D6 (0.34) GRIN2BGRIN1CYP2D6HRH1KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1664059-B1 THIENOPYRROLES AS ANTIVIRAL AGENTS ANGELETTI P IST RICHERCHE BIO (IT) 2007-09-12 EP claimed