SCHEMBL5228879

SCHEMBL5228879

O=C(c1ccccc1)C1CCCN(Cc2cnn(-c3ccc(-c4ccc(F)cc4)cc3)c2-c2ccco2)C1

nearest known ligand 0.47

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 4/20 0.47
ALDH1A1 P00352 2/20 0.47
MAPK1 P28482 2/20 0.47
MEN1 O00255 2/20 0.47
NPC1 O15118 1/20 0.47
RAB9A P51151 1/20 0.47
BLM P54132 1/20 0.47
MAPT P10636 1/20 0.46
LMNA P02545 2/20 0.45
KDM2B Q8NHM5 4/20 0.44
CYP1A2 P05177 1/20 0.43
CYP3A4 P08684 1/20 0.43
CYP2C9 P11712 1/20 0.43
RECQL P46063 1/20 0.42
TDP1 Q9NUW8 1/20 0.42
KDM4E B2RXH2 1/20 0.41
POLB P06746 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5228002 0.85 TSHR (0.39) KMT2AALDH1A1NPC1KDM4EPOLB
SCHEMBL5225875 0.80 CYP2D6 (0.36) ALDH1A1MAPTCYP3A4CYP2C9POLB
SCHEMBL5223970 0.78 ADORA2A (0.40) ALDH1A1MAPTLMNA
SCHEMBL5222786 0.77 GRM2 (0.38) KDM4E
SCHEMBL2761177 0.77 DRD4 (0.42) KMT2AALDH1A1MEN1MAPTKDM4E
SCHEMBL2761237 0.76 SMO (0.43) ALDH1A1MAPTLMNAKDM4E
SCHEMBL2761009 0.76 SMO (0.43) ALDH1A1MAPTLMNA
Hydrochloric Acid SCHEMBL1997589 0.75 SMO (0.42) ALDH1A1MAPTLMNAKDM4E
SCHEMBL5228047 0.74 HTR2C (0.37) ALDH1A1KDM4E
SCHEMBL2761137 0.73 SMO (0.41) KMT2AALDH1A1MAPTLMNAPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1611122-B1 SUBSTITUTED PYRAZOLE COMPOUNDS MERCK PATENT GMBH (DE) 2007-06-13 EP disclosed