SCHEMBL5229004

SCHEMBL5229004

COc1ccc(-c2ccc(-n3ncc(CN(Cc4nccn4C)Cc4nccn4C)c3-c3ccco3)cc2)cc1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPBWR1 P48145 2/20 0.40
MCHR1 Q99705 1/20 0.40
PTGS1 P23219 1/20 0.38
PTGS2 P35354 1/20 0.38
TP53 P04637 3/20 0.37
KDM4E B2RXH2 3/20 0.37
MAPT P10636 2/20 0.36
HPGD P15428 2/20 0.36
HSD17B10 Q99714 2/20 0.36
NPC1 O15118 1/20 0.36
RAB9A P51151 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
NPSR1 Q6W5P4 1/20 0.34
ADORA2A P29274 1/20 0.34
ALDH1A1 P00352 3/20 0.34
TSHR P16473 1/20 0.34
SIRT1 Q96EB6 1/20 0.34
TUBB4A P04350 1/20 0.34
TUBB P07437 1/20 0.34
TUBA3C P0DPH7 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5224717 0.84 NPBWR1 (0.45) NPBWR1MCHR1PTGS1PTGS2TP53
SCHEMBL5226619 0.82 NPBWR1 (0.47) NPBWR1MCHR1PTGS1PTGS2TP53
SCHEMBL5228410 0.78 PTGS1 (0.49) NPBWR1MCHR1PTGS1PTGS2TP53
SCHEMBL5224302 0.74 SMO (0.49) NPBWR1MCHR1PTGS1PTGS2TP53
SCHEMBL5232263 0.74 SMO (0.49) NPBWR1MCHR1PTGS1PTGS2TP53
SCHEMBL5230237 0.73 MAPT (0.47) NPBWR1MCHR1PTGS1PTGS2TP53
SCHEMBL5230220 0.73 NPBWR1 (0.40) NPBWR1MCHR1PTGS1PTGS2TP53
SCHEMBL5230456 0.72 SMO (0.46) NPBWR1MCHR1PTGS1PTGS2TP53
SCHEMBL5225666 0.72 NPBWR1 (0.43) NPBWR1MCHR1PTGS1PTGS2TP53
SCHEMBL5226649 0.70 F10 (0.41) NPBWR1MCHR1TP53KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1611122-B1 SUBSTITUTED PYRAZOLE COMPOUNDS MERCK PATENT GMBH (DE) 2007-06-13 EP disclosed