SCHEMBL5229628

SCHEMBL5229628

COC(=O)Oc1cc2c([N+](=O)[O-])cccc2s1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC9A1 P19634 2/20 0.53
ALDH1A1 P00352 4/20 0.43
MEN1 O00255 2/20 0.41
KMT2A Q03164 2/20 0.41
POLB P06746 1/20 0.41
TDP1 Q9NUW8 1/20 0.41
TSHR P16473 1/20 0.39
NPSR1 Q6W5P4 2/20 0.39
MAPT P10636 1/20 0.39
AKR1C4 P17516 1/20 0.39
AKR1C3 P42330 1/20 0.39
AKR1C2 P52895 1/20 0.39
AKR1C1 Q04828 1/20 0.39
GLA P06280 1/20 0.39
LMNA P02545 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
RAB9A P51151 1/20 0.38
HDAC3 O15379 1/20 0.37
HDAC4 P56524 1/20 0.37
HDAC1 Q13547 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5230549 0.86 SLC9A1 (0.52) SLC9A1ALDH1A1MEN1KMT2APOLB
SCHEMBL5231955 0.82 MEN1 (0.51) SLC9A1ALDH1A1MEN1KMT2APOLB
SCHEMBL5231463 0.80 SLC9A1 (0.47) SLC9A1ALDH1A1MEN1KMT2APOLB
SCHEMBL829093 0.80 SLC9A1 (0.61) SLC9A1ALDH1A1MEN1KMT2APOLB
SCHEMBL8187301 0.74 ALDH1A1 (0.37) ALDH1A1MAPTLMNA
SCHEMBL5202332 0.74 SMN1; SMN2 (0.49) ALDH1A1MEN1KMT2APOLBTDP1
SCHEMBL5231561 0.74 SMN1; SMN2 (0.62) ALDH1A1MEN1KMT2APOLBTDP1
SCHEMBL5198179 0.73 HDAC3 (0.49) SLC9A1LMNARAB9AHDAC3HDAC4
SCHEMBL2893474 0.73 SLC9A1 (0.67) SLC9A1ALDH1A1MEN1KMT2APOLB
SCHEMBL7448258 0.72 SMN1; SMN2 (0.47) ALDH1A1MEN1KMT2APOLBTDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1461335-B1 2-HETEROARYLCARBOXYLIC ACID AMIDES BAYER HEALTHCARE AG (DE) 2007-02-28 EP disclosed
EP-1461335-A1 2-HETEROARYLCARBOXYLIC ACID AMIDES Bayer HealthCare AG (DE) 2004-09-29 EP disclosed
WO-2003055878-A1 2-HETEROARYLCARBOXYLIC ACID AMIDES BAYER HEALTHCARE AG (DE) 2003-07-10 WO disclosed