SCHEMBL5229977

SCHEMBL5229977

CN(C)Cc1c(OC(=O)O)sc2c(C3CCCCC3)c(-c3ccc(Cl)cc3)n(C)c12

nearest known ligand 0.38

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CNR1 P21554 4/20 0.36
CYP3A4 P08684 1/20 0.33
CYP2C19 P33261 1/20 0.33
TACR1 P25103 2/20 0.33
PTGDR Q13258 2/20 0.32
PTGDR2 Q9Y5Y4 2/20 0.32
PTGER2 P43116 1/20 0.32
TP53 P04637 1/20 0.32
MAPT P10636 1/20 0.32
AGER Q15109 1/20 0.31
HRH3 Q9Y5N1 1/20 0.31
PROKR1 Q8TCW9 1/20 0.31
LSS P48449 1/20 0.31
ALDH1A1 P00352 1/20 0.31
SLC6A9 P48067 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2997212 0.87 CNR1 (0.37) CNR1CYP3A4CYP2C19TACR1TP53
SCHEMBL5231069 0.86 LSS (0.36) CNR1TACR1HRH3LSSALDH1A1
SCHEMBL5230079 0.85 MMP2 (0.35) CNR1CYP3A4CYP2C19TACR1
SCHEMBL5233254 0.85 TACR1 (0.36) CNR1CYP3A4CYP2C19TACR1TP53
SCHEMBL5227454 0.83 ALDH1A1 (0.34) CNR1TACR1ALDH1A1
SCHEMBL5228235 0.82 EGFR (0.39) TACR1TP53MAPTALDH1A1
SCHEMBL5234741 0.81 CNR1 (0.34) CNR1CYP3A4CYP2C19TP53MAPT
SCHEMBL5227012 0.77 CYP3A4 (0.40) CNR1CYP3A4CYP2C19TACR1PTGDR
SCHEMBL3001005 0.75 MEN1 (0.36) CNR1TACR1HRH3ALDH1A1
SCHEMBL2996688 0.74 MMP2 (0.35) CNR1CYP3A4CYP2C19TACR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1664059-B1 THIENOPYRROLES AS ANTIVIRAL AGENTS ANGELETTI P IST RICHERCHE BIO (IT) 2007-09-12 EP claimed