SCHEMBL5231609

SCHEMBL5231609

Cc1noc(C)c1C(=O)N1CC2CN(c3cccc(CCC(N)=O)c3)CC2C1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 7/20 0.48
USP2 O75604 5/20 0.48
ALDH1A1 P00352 4/20 0.48
HSD17B10 Q99714 2/20 0.48
HIF1A Q16665 2/20 0.48
MAPK1 P28482 2/20 0.47
HPGD P15428 2/20 0.47
LMNA P02545 1/20 0.44
CYP3A4 P08684 5/20 0.44
TSHR P16473 4/20 0.44
CYP2D6 P10635 3/20 0.44
CYP1A2 P05177 2/20 0.44
ALOX15 P16050 1/20 0.44
MAPT P10636 1/20 0.44
CCR5 P51681 1/20 0.42
CYP2C9 P11712 3/20 0.42
MEN1 O00255 3/20 0.41
KMT2A Q03164 3/20 0.41
KDM4E B2RXH2 1/20 0.41
CYP2C19 P33261 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5229641 0.88 LMNA (0.53) SMN1; SMN2USP2ALDH1A1HSD17B10HIF1A
SCHEMBL4968486 0.85 HCRTR1 (0.42) CCR5HCRTR1HCRTR2
SCHEMBL4692413 0.85 HCRTR1 (0.53) CCR5HCRTR1HCRTR2
SCHEMBL5235800 0.83 HCRTR1 (0.44) CCR5HCRTR1HCRTR2
SCHEMBL5233360 0.83 HTT (0.47) SMN1; SMN2USP2MAPK1LMNATSHR
SCHEMBL5230484 0.83 HCRTR1 (0.44) HCRTR1HCRTR2
SCHEMBL4698184 0.82 HCRTR1 (0.46) HCRTR1HCRTR2
SCHEMBL4809142 0.82 HCRTR1 (0.41) USP2MAPTHCRTR1HCRTR2
SCHEMBL4699432 0.82 CCL5 (0.44) SMN1; SMN2USP2ALDH1A1LMNACYP3A4
SCHEMBL5236364 0.82 HCRTR1 (0.47) CCR5HCRTR1HCRTR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1761542-A2 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS F.HOFFMANN-LA ROCHE AG (CH) 2007-03-14 EP claimed
WO-2005121145-A2 OCTAHYDRO-PYRROLO[3,4-C] DERIVATIVES AND THEIR USE AS ANTIVIRAL COMPOUNDS F. HOFFMANN-LA ROCHE AG (CH) 2005-12-22 WO claimed