SCHEMBL5232859

SCHEMBL5232859

CSCC(=O)NCCCc1cccc(N2CC3CN(C(=O)c4c(F)cccc4Cl)CC3C2)c1

nearest known ligand 0.40

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
HCRTR1 O43613 10/20 0.40
HCRTR2 O43614 10/20 0.40
SIGMAR1 Q99720 1/20 0.38
LMNA P02545 1/20 0.37
MAPK1 P28482 1/20 0.37
GAA P10253 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5233381 0.89 HCRTR1 (0.41) HCRTR1HCRTR2SIGMAR1
SCHEMBL5233744 0.89 ALDH1A1 (0.41) HCRTR1HCRTR2SIGMAR1LMNA
SCHEMBL5237863 0.89 SIGMAR1 (0.41) HCRTR1HCRTR2SIGMAR1LMNA
SCHEMBL5234742 0.89 HCRTR1 (0.40) HCRTR1HCRTR2SIGMAR1
SCHEMBL5235325 0.89 HCRTR1 (0.40) HCRTR1HCRTR2SIGMAR1LMNA
SCHEMBL5237039 0.89 HCRTR1 (0.40) HCRTR1HCRTR2SIGMAR1
SCHEMBL5236854 0.88 HPGD (0.43) HCRTR1HCRTR2SIGMAR1GAA
SCHEMBL5233648 0.88 HCRTR1 (0.42) HCRTR1HCRTR2SIGMAR1LMNA
SCHEMBL5237363 0.88 HCRTR1 (0.39) HCRTR1HCRTR2SIGMAR1LMNA
SCHEMBL5235332 0.87 HCRTR1 (0.42) HCRTR1HCRTR2SIGMAR1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1761542-A2 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS F.HOFFMANN-LA ROCHE AG (CH) 2007-03-14 EP claimed
WO-2005121145-A2 OCTAHYDRO-PYRROLO[3,4-C] DERIVATIVES AND THEIR USE AS ANTIVIRAL COMPOUNDS F. HOFFMANN-LA ROCHE AG (CH) 2005-12-22 WO claimed