SCHEMBL5237863

SCHEMBL5237863

NCCC(=O)NCCCc1cccc(N2CC3CN(C(=O)c4c(F)cccc4Cl)CC3C2)c1

nearest known ligand 0.41

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 1/20 0.41
HCRTR1 O43613 7/20 0.40
HCRTR2 O43614 7/20 0.40
MAPK8 P45983 1/20 0.37
MAPK10 P53779 1/20 0.37
HPGD P15428 1/20 0.36
MGLL Q99685 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.35
ALDH1A1 P00352 1/20 0.35
LMNA P02545 1/20 0.35
TSHR P16473 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5238559 0.94 SIGMAR1 (0.40) SIGMAR1HCRTR1HCRTR2MAPK8MAPK10
SCHEMBL5236854 0.91 HPGD (0.43) SIGMAR1HCRTR1HCRTR2MAPK8MAPK10
SCHEMBL5233648 0.90 HCRTR1 (0.42) SIGMAR1HCRTR1HCRTR2MAPK8MAPK10
SCHEMBL5236149 0.90 MAPK1 (0.40) SIGMAR1HCRTR1HCRTR2L3MBTL1ALDH1A1
SCHEMBL5233744 0.90 ALDH1A1 (0.41) SIGMAR1HCRTR1HCRTR2HPGDALDH1A1
SCHEMBL5233381 0.90 HCRTR1 (0.41) SIGMAR1HCRTR1HCRTR2
SCHEMBL5237363 0.90 HCRTR1 (0.39) SIGMAR1HCRTR1HCRTR2MAPK8MAPK10
SCHEMBL5234646 0.90 HCRTR1 (0.38) SIGMAR1HCRTR1HCRTR2HPGD
SCHEMBL5238325 0.90 GAA (0.39) SIGMAR1HCRTR1HCRTR2
SCHEMBL5235733 0.90 SIGMAR1 (0.44) SIGMAR1HCRTR1HCRTR2MAPK8MAPK10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1761542-A2 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS F.HOFFMANN-LA ROCHE AG (CH) 2007-03-14 EP claimed
WO-2005121145-A2 OCTAHYDRO-PYRROLO[3,4-C] DERIVATIVES AND THEIR USE AS ANTIVIRAL COMPOUNDS F. HOFFMANN-LA ROCHE AG (CH) 2005-12-22 WO claimed