SCHEMBL5233869

SCHEMBL5233869

CCNC(=O)N1CCC(N(c2nn(-c3ccccc3)cc2OC(=O)O)C(=O)[C@H]2CC[C@H](C)CC2)CC1

nearest known ligand 0.36

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
OPRM1 P35372 5/20 0.36
GAA P10253 2/20 0.35
BRD4 O60885 1/20 0.35
CHRM2 P08172 1/20 0.34
CHRM3 P20309 1/20 0.34
CACNA2D1 P54289 2/20 0.33
USP2 O75604 1/20 0.33
ATM Q13315 1/20 0.33
KMT2A Q03164 1/20 0.33
CDK1 P06493 1/20 0.33
CDK4 P11802 1/20 0.33
CCND1 P24385 1/20 0.33
CDK2 P24941 1/20 0.33
OPRD1 P41143 1/20 0.33
POLB P06746 1/20 0.33
NPSR1 Q6W5P4 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5232559 0.88 OPRM1 (0.37) OPRM1GAABRD4CHRM2CHRM3
SCHEMBL5232570 0.88 OPRM1 (0.37) OPRM1GAABRD4CHRM2CHRM3
SCHEMBL5234101 0.88 GAA (0.39) OPRM1GAABRD4CACNA2D1USP2
SCHEMBL5236494 0.88 GAA (0.35) OPRM1GAACHRM2CHRM3CACNA2D1
SCHEMBL5239704 0.86 NPSR1 (0.41) OPRM1GAABRD4USP2ATM
SCHEMBL5239714 0.86 NPSR1 (0.41) OPRM1GAABRD4USP2ATM
SCHEMBL5237036 0.86 CACNA2D1 (0.42) OPRM1CHRM2CHRM3CACNA2D1POLB
SCHEMBL5237215 0.85 CACNA2D1 (0.36) OPRM1CHRM2CHRM3CACNA2D1KMT2A
SCHEMBL5237690 0.84 CACNA2D1 (0.41) OPRM1CACNA2D1KMT2A
SCHEMBL5238148 0.83 POLB (0.40) OPRM1CACNA2D1POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1730116-B1 4-CARBOX PYRAZOLE DERIVATES USEFUL AS ANTI-VIRAL AGENTS SMITHKLINE BEECHAM CORP (US) 2007-09-05 EP claimed