SCHEMBL5234101

SCHEMBL5234101

COC(=O)N1CCC(N(c2nn(-c3ccccc3)cc2OC(=O)O)C(=O)[C@H]2CC[C@H](C)CC2)CC1

nearest known ligand 0.39

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
GAA P10253 2/20 0.39
KMT2A Q03164 5/20 0.35
MEN1 O00255 4/20 0.35
CYP3A4 P08684 2/20 0.35
CYP2C19 P33261 2/20 0.35
NPC1 O15118 2/20 0.35
RAB9A P51151 2/20 0.35
MAPK1 P28482 1/20 0.35
USP2 O75604 1/20 0.34
HSD17B10 Q99714 1/20 0.34
BRD4 O60885 1/20 0.34
OPRM1 P35372 3/20 0.34
GPR119 Q8TDV5 1/20 0.33
CACNA2D1 P54289 3/20 0.33
KDM4E B2RXH2 1/20 0.33
ALDH1A1 P00352 1/20 0.33
POLB P06746 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5236494 0.91 GAA (0.35) GAAUSP2OPRM1CACNA2D1ALDH1A1
SCHEMBL5237036 0.89 CACNA2D1 (0.42) OPRM1CACNA2D1KDM4EALDH1A1POLB
SCHEMBL5231976 0.88 ATM (0.37) GAAKMT2AMEN1CYP3A4CYP2C19
SCHEMBL5231969 0.88 ATM (0.37) GAAKMT2AMEN1CYP3A4CYP2C19
SCHEMBL5233869 0.88 OPRM1 (0.36) GAAKMT2AUSP2BRD4OPRM1
SCHEMBL5237215 0.88 CACNA2D1 (0.36) KMT2AMEN1NPC1RAB9AOPRM1
SCHEMBL5238148 0.86 POLB (0.40) OPRM1CACNA2D1KDM4EALDH1A1POLB
SCHEMBL5237690 0.85 CACNA2D1 (0.41) KMT2AMEN1NPC1RAB9AOPRM1
SCHEMBL5235781 0.85 ALDH1A1 (0.34) GAAKMT2AMEN1NPC1RAB9A
SCHEMBL5233912 0.84 KDM4E (0.42) GAAKMT2ANPC1RAB9AMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1730116-B1 4-CARBOX PYRAZOLE DERIVATES USEFUL AS ANTI-VIRAL AGENTS SMITHKLINE BEECHAM CORP (US) 2007-09-05 EP claimed