SCHEMBL5237690

SCHEMBL5237690

C[C@H]1CC[C@H](C(=O)N(c2nn(-c3ccccc3)cc2OC(=O)O)C2CCNCC2)CC1

nearest known ligand 0.41

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CACNA2D1 P54289 5/20 0.41
KHK P50053 4/20 0.34
KMT2A Q03164 2/20 0.33
NPC1 O15118 2/20 0.33
RAB9A P51151 2/20 0.33
MEN1 O00255 1/20 0.33
KCNH2 Q12809 2/20 0.33
UCHL1 P09936 1/20 0.32
OPRM1 P35372 3/20 0.31
DRD4 P21917 1/20 0.31
PARP1 P09874 1/20 0.31
SLC6A2 P23975 1/20 0.31
SLC6A4 P31645 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5237215 0.91 CACNA2D1 (0.36) CACNA2D1KMT2ANPC1RAB9AMEN1
SCHEMBL5237036 0.89 CACNA2D1 (0.42) CACNA2D1OPRM1
SCHEMBL5235781 0.89 ALDH1A1 (0.34) CACNA2D1KMT2ANPC1RAB9AMEN1
SCHEMBL5236494 0.87 GAA (0.35) CACNA2D1UCHL1OPRM1
SCHEMBL5230826 0.86 CACNA2D1 (0.42) CACNA2D1KHKKMT2AMEN1KCNH2
SCHEMBL5230831 0.86 CACNA2D1 (0.42) CACNA2D1KHKKMT2AMEN1KCNH2
SCHEMBL5234101 0.85 GAA (0.39) CACNA2D1KMT2ANPC1RAB9AMEN1
SCHEMBL5238148 0.85 POLB (0.40) CACNA2D1OPRM1
SCHEMBL5233869 0.84 OPRM1 (0.36) CACNA2D1KMT2AOPRM1
SCHEMBL5231854 0.83 NPSR1 (0.44) CACNA2D1NPC1RAB9ADRD4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1730116-B1 4-CARBOX PYRAZOLE DERIVATES USEFUL AS ANTI-VIRAL AGENTS SMITHKLINE BEECHAM CORP (US) 2007-09-05 EP claimed