SCHEMBL5236494

SCHEMBL5236494

CC(=O)N1CCC(N(c2nn(-c3ccccc3)cc2OC(=O)O)C(=O)[C@H]2CC[C@H](C)CC2)CC1

nearest known ligand 0.35

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
GAA P10253 1/20 0.35
ALDH1A1 P00352 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.34
OPRM1 P35372 7/20 0.34
CACNA2D1 P54289 5/20 0.34
NPY5R Q15761 1/20 0.33
UCHL1 P09936 1/20 0.33
CHRM2 P08172 1/20 0.33
CHRM3 P20309 1/20 0.33
ACHE P22303 1/20 0.33
USP2 O75604 1/20 0.33
ATM Q13315 1/20 0.33
RIPK1 Q13546 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5234101 0.91 GAA (0.39) GAAALDH1A1OPRM1CACNA2D1USP2
SCHEMBL5237036 0.91 CACNA2D1 (0.42) ALDH1A1OPRM1CACNA2D1CHRM2CHRM3
SCHEMBL5237215 0.89 CACNA2D1 (0.36) ALDH1A1OPRM1CACNA2D1UCHL1CHRM2
SCHEMBL5233869 0.88 OPRM1 (0.36) GAAOPRM1CACNA2D1CHRM2CHRM3
SCHEMBL5238148 0.87 POLB (0.40) ALDH1A1L3MBTL1OPRM1CACNA2D1NPY5R
SCHEMBL5237690 0.87 CACNA2D1 (0.41) OPRM1CACNA2D1UCHL1
SCHEMBL5235781 0.87 ALDH1A1 (0.34) GAAALDH1A1L3MBTL1OPRM1CACNA2D1
SCHEMBL5235207 0.87 L3MBTL1 (0.35) ALDH1A1L3MBTL1OPRM1CACNA2D1NPY5R
SCHEMBL5235195 0.87 L3MBTL1 (0.35) ALDH1A1L3MBTL1OPRM1CACNA2D1NPY5R
SCHEMBL5232225 0.83 NPSR1 (0.43) ALDH1A1L3MBTL1OPRM1CACNA2D1USP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1730116-B1 4-CARBOX PYRAZOLE DERIVATES USEFUL AS ANTI-VIRAL AGENTS SMITHKLINE BEECHAM CORP (US) 2007-09-05 EP claimed