SCHEMBL5236254

SCHEMBL5236254

N#Cc1cccc(C(=O)N2CC3CN(c4cccc(CCC(N)=O)c4)CC3C2)c1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PLA2G10 O15496 1/20 0.41
PLA2G2A P14555 1/20 0.41
HTR7 P34969 1/20 0.41
TMEM97 Q5BJF2 1/20 0.41
NOTUM Q6P988 1/20 0.40
NAMPT P43490 2/20 0.38
CHRM4 P08173 2/20 0.38
GRM5 P41594 2/20 0.38
CYP3A4 P08684 1/20 0.38
CYP2C9 P11712 1/20 0.38
SLC9A1 P19634 1/20 0.38
CYP2C19 P33261 1/20 0.38
SIRT2 Q8IXJ6 1/20 0.37
SIRT1 Q96EB6 1/20 0.37
GSK3B P49841 1/20 0.36
NOS2 P35228 1/20 0.36
KCNJ1 P48048 1/20 0.36
KCNH2 Q12809 1/20 0.36
PARP1 P09874 1/20 0.36
FFAR1 O14842 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5236638 0.91 ALDH1A1 (0.44) PLA2G10PLA2G2AHTR7TMEM97CYP3A4
SCHEMBL5232788 0.87 CHRNB2 (0.44) PLA2G10PLA2G2AKCNH2
SCHEMBL4694475 0.85 SMN1; SMN2 (0.47) CYP3A4CYP2C9CYP2C19
SCHEMBL5238361 0.85 HPGD (0.43) PLA2G10HTR7PARP1
SCHEMBL5234579 0.85 HCRTR1 (0.42) PLA2G10PLA2G2AHTR7TMEM97NOTUM
SCHEMBL5233538 0.82 ALDH1A1 (0.47) PLA2G10
SCHEMBL4694593 0.82 ALDH1A1 (0.41) PLA2G10PLA2G2AHTR7
SCHEMBL5230954 0.81 GABRD (0.42) NAMPTSIRT1
SCHEMBL5235769 0.80 CHRNA4 (0.47) PLA2G10PLA2G2ANAMPT
SCHEMBL5235877 0.79 ALDH1A1 (0.48) CYP3A4CYP2C9CYP2C19PARP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1761542-A2 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS F.HOFFMANN-LA ROCHE AG (CH) 2007-03-14 EP claimed
WO-2005121145-A2 OCTAHYDRO-PYRROLO[3,4-C] DERIVATIVES AND THEIR USE AS ANTIVIRAL COMPOUNDS F. HOFFMANN-LA ROCHE AG (CH) 2005-12-22 WO claimed