SCHEMBL5236342

SCHEMBL5236342

CC(C)N(c1nn(-c2ccc(OC(F)(F)F)cc2)cc1OC(=O)O)C(=O)[C@H]1CC[C@H](C)CC1

nearest known ligand 0.38

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
CHRM4 P08173 4/20 0.38
EPHX2 P34913 2/20 0.36
LIPE Q05469 5/20 0.35
GCGR P47871 1/20 0.34
GIPR P48546 1/20 0.34
IDH1 O75874 4/20 0.33
PTGDR2 Q9Y5Y4 1/20 0.33
PPARD Q03181 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5236675 0.91 NOTUM (0.40) CHRM4
SCHEMBL5231923 0.89 TRPA1 (0.35) LIPEPTGDR2
SCHEMBL5234129 0.89 ADORA3 (0.37)
SCHEMBL5228551 0.88 CHRM4 (0.39) CHRM4EPHX2LIPEGCGRGIPR
SCHEMBL5228545 0.88 CHRM4 (0.39) CHRM4EPHX2LIPEGCGRGIPR
SCHEMBL5234466 0.87 APP (0.36)
SCHEMBL5236797 0.87
SCHEMBL5236128 0.87 NPC1 (0.34)
SCHEMBL5233446 0.87 NPC1 (0.35)
SCHEMBL5232338 0.86 S1PR1 (0.34)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1730116-B1 4-CARBOX PYRAZOLE DERIVATES USEFUL AS ANTI-VIRAL AGENTS SMITHKLINE BEECHAM CORP (US) 2007-09-05 EP claimed