SCHEMBL5236506

SCHEMBL5236506

CC(C)N(c1nn(-c2ccc(OCc3cscn3)cc2)cc1OC(=O)O)C(=O)[C@H]1CC[C@H](C)CC1

nearest known ligand 0.41

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
ALOX5 P09917 1/20 0.41
MMP13 P45452 1/20 0.33
MMP14 P50281 1/20 0.33
MAPK14 Q16539 1/20 0.31
ALDH1A1 P00352 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5236497 0.90 ALOX5 (0.41) ALOX5MMP13MMP14MAPK14ALDH1A1
SCHEMBL5238294 0.90 ALOX5 (0.41) ALOX5MMP13MMP14MAPK14ALDH1A1
SCHEMBL5233481 0.89 ALDH1A1 (0.30) ALOX5ALDH1A1
SCHEMBL5236015 0.86 KDM4E (0.43) ALDH1A1
SCHEMBL5236069 0.85 ALOX5 (0.38) ALOX5MMP13MMP14MAPK14ALDH1A1
SCHEMBL5236077 0.85 ALOX5 (0.38) ALOX5MMP13MMP14MAPK14ALDH1A1
SCHEMBL5236387 0.85 KDM4E (0.39) ALDH1A1
SCHEMBL5234129 0.83 ADORA3 (0.37) ALDH1A1
SCHEMBL5236797 0.83
SCHEMBL5236283 0.83

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1730116-B1 4-CARBOX PYRAZOLE DERIVATES USEFUL AS ANTI-VIRAL AGENTS SMITHKLINE BEECHAM CORP (US) 2007-09-05 EP claimed