SCHEMBL5238526

SCHEMBL5238526

CNC1(CC=O)CN(c2ccc(C)cn2)CCN1C(=O)O

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PANK3 Q9H999 1/20 0.39
PPARG P37231 1/20 0.37
PPARA Q07869 1/20 0.37
RAB9A P51151 2/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
PARP1 P09874 1/20 0.35
HDAC1 Q13547 2/20 0.34
GRIN2D O15399 1/20 0.34
GRIN3B O60391 1/20 0.34
GRIN1 Q05586 1/20 0.34
GRIN2A Q12879 1/20 0.34
GRIN2B Q13224 1/20 0.34
GRIN2C Q14957 1/20 0.34
GRIN3A Q8TCU5 1/20 0.34
DHFR P00374 1/20 0.34
AOC3 Q16853 1/20 0.34
DRD2 P14416 2/20 0.33
DRD1 P21728 2/20 0.33
DRD5 P21918 2/20 0.33
DRD3 P35462 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5237945 0.90 PANK3 (0.37) PANK3PPARGPPARARAB9AL3MBTL1
SCHEMBL5233815 0.86 PANK3 (0.35) PANK3PPARGPPARARAB9AL3MBTL1
SCHEMBL5237467 0.85 PANK3 (0.40) PANK3HDAC1AOC3KMT2AHRH3
SCHEMBL5236758 0.85 EGLN1 (0.40) PANK3RAB9ADRD2
SCHEMBL5235197 0.84 HSD17B10 (0.45) CYP1A2CYP2C19HTR1AMAPTCYP2C9
SCHEMBL5239788 0.83 MAPT (0.43) RAB9AL3MBTL1CYP2C19KMT2AMAPT
SCHEMBL5238354 0.83 MAPT (0.40) CYP1A2CYP2C19KMT2AMAPTMEN1
SCHEMBL5233798 0.82 AKR1C3 (0.36) PANK3PPARGPPARARAB9AHDAC1
SCHEMBL5231485 0.82 HTR3A (0.44) HDAC1DRD2DRD3HTR1AHTR2A
SCHEMBL5237297 0.82 KDM4E (0.40) L3MBTL1HRH3MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1701946-B1 DERIVATIVES OF 1-PIPERAZINE- AND 1-HOMOPIPERAZINE-CARBOXYLATES, PREPARATION METHOD THEREOF AND USE OF SAME AS INHIBITORS OF THE FAAH ENZYME SANOFI AVENTIS (FR) 2007-12-19 EP claimed