SCHEMBL5235197

SCHEMBL5235197

CNC1(CC=O)CN(c2ccccn2)CCN1C(=O)O

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSD17B10 Q99714 7/20 0.45
KDM4E B2RXH2 6/20 0.45
HPGD P15428 5/20 0.45
CYP2C9 P11712 3/20 0.45
CYP3A4 P08684 3/20 0.45
RECQL P46063 1/20 0.45
THRB P10828 1/20 0.42
NPSR1 Q6W5P4 1/20 0.42
ALDH1A1 P00352 8/20 0.42
CYP2D6 P10635 4/20 0.42
POLB P06746 2/20 0.42
TSHR P16473 4/20 0.41
USP2 O75604 1/20 0.41
HIF1A Q16665 1/20 0.41
CYP2C19 P33261 3/20 0.41
CYP1A2 P05177 2/20 0.41
MAPK1 P28482 1/20 0.41
HTR1A P08908 1/20 0.41
BCHE P06276 1/20 0.40
ACHE P22303 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5237297 0.85 KDM4E (0.40) KDM4ETHRBALDH1A1MAPT
SCHEMBL5238192 0.84 CYP2C19 (0.37) HSD17B10CYP2C9CYP3A4NPSR1ALDH1A1
SCHEMBL5238526 0.84 PANK3 (0.39) CYP2C9CYP2C19CYP1A2HTR1AMAPT
SCHEMBL5231485 0.83 HTR3A (0.44) ALDH1A1TSHRHTR1A
SCHEMBL5238157 0.82 KDM4E (0.48) HSD17B10KDM4EHPGDCYP3A4RECQL
SCHEMBL5236555 0.80 USP2 (0.41) HSD17B10HPGDCYP2C9CYP3A4ALDH1A1
SCHEMBL5235916 0.80 AR (0.40) KDM4ECYP2C9ALDH1A1TSHRCYP2C19
SCHEMBL5237871 0.80 DRD2 (0.40) ALDH1A1HTR1AMAPT
SCHEMBL5238575 0.78 CXCR3 (0.38) HTR1A
SCHEMBL5238354 0.78 MAPT (0.40) KDM4EHPGDCYP2C9CYP3A4ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1701946-B1 DERIVATIVES OF 1-PIPERAZINE- AND 1-HOMOPIPERAZINE-CARBOXYLATES, PREPARATION METHOD THEREOF AND USE OF SAME AS INHIBITORS OF THE FAAH ENZYME SANOFI AVENTIS (FR) 2007-12-19 EP claimed